SCHEMBL4011017

SCHEMBL4011017

CCCc1nc(CCF)c(Cc2ccc(-c3ccccc3C#N)cc2)c(=O)[nH]1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PPARG P37231 2/20 0.43
ACHE P22303 1/20 0.39
AGTR1 P30556 2/20 0.38
PRMT5 O14744 1/20 0.37
WDR77 Q9BQA1 1/20 0.37
PDE3B Q13370 1/20 0.37
PDE3A Q14432 1/20 0.37
BRS3 P32247 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1894561 0.91 ACHE (0.45) PPARGACHEAGTR1PDE3BPDE3A
SCHEMBL1886733 0.89 PPARG (0.45) PPARGACHEAGTR1
SCHEMBL4011221 0.87 PPARG (0.43) PPARGACHEAGTR1PDE3BPDE3A
SCHEMBL12348665 0.85 ACHE (0.45) PPARGACHEAGTR1
SCHEMBL1886429 0.85 ACHE (0.43) PPARGACHEAGTR1BRS3
SCHEMBL1892195 0.84 ACHE (0.44) PPARGACHEAGTR1
SCHEMBL4013842 0.84 PPARG (0.43) PPARGACHEAGTR1PDE3BPDE3A
SCHEMBL4312700 0.84 PPARG (0.43) PPARGACHEAGTR1PDE3BPDE3A
SCHEMBL4016051 0.84 ACHE (0.43) PPARGACHEAGTR1
SCHEMBL1896983 0.84 PPARG (0.46) PPARGACHEAGTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009133970-A1 CRYSTALLINE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-11-05 WO disclosed
EP-2074117-A2 HETEROMONOCYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2009-07-01 EP disclosed
WO-2008062905-A2 HETEROMONOCYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-05-29 WO disclosed