SCHEMBL401110

SCHEMBL401110

Clc1ccc2c(Cl)ncnc2c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.57
PDE4B Q07343 1/20 0.57
PDE4C Q08493 1/20 0.57
PDE4D Q08499 1/20 0.57
NR4A2 P43354 1/20 0.50
SOS2 Q07890 1/20 0.50
CYP1A2 P05177 2/20 0.47
CYP2D6 P10635 1/20 0.47
ALDH1A1 P00352 3/20 0.47
LMNA P02545 3/20 0.46
KMT2A Q03164 3/20 0.46
GPR55 Q9Y2T6 1/20 0.46
KDM4E B2RXH2 1/20 0.45
HPGD P15428 1/20 0.45
HTT P42858 3/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
MEN1 O00255 1/20 0.44
PPARG P37231 1/20 0.44
RXFP1 Q9HBX9 1/20 0.44
NR2E3 Q9Y5X4 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29416410 1.00 PDE4A (0.57) PDE4APDE4BPDE4CPDE4DNR4A2
Hydrochloric Acid SCHEMBL5739823 0.98 PDE4A (0.55) PDE4APDE4BPDE4CPDE4DNR4A2
SCHEMBL856909 0.83 PDE4A (0.57) PDE4APDE4BPDE4CPDE4DNR4A2
SCHEMBL29793572 0.83 PDE4A (0.57) PDE4APDE4BPDE4CPDE4DNR4A2
SCHEMBL145141 0.79 PDE4A (0.53) PDE4APDE4BPDE4CPDE4DCYP1A2
SCHEMBL856547 0.79 PDE4A (0.53) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL20813787 0.79 NR4A2 (0.47) NR4A2SOS2CYP1A2CYP2D6ALDH1A1
SCHEMBL22911854 0.79 PDE4A (0.53) PDE4APDE4BPDE4CPDE4DNR4A2
SCHEMBL858150 0.79 PDE4A (0.53) PDE4APDE4BPDE4CPDE4DCYP1A2
SCHEMBL6442231 0.79 NR4A2 (0.56) NR4A2SOS2CYP1A2CYP2D6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 310 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114105892-B FAK/PLK1 double-target quinazoline derivative and preparation method and application thereof 浙江科技学院 2024-03-26 CN claimed
CN-114105892-A FAK/PLK1 dual-target quinazoline derivative and preparation method and application thereof 浙江科技学院 2022-03-01 CN claimed
JP-59013765-A None JP disclosed
EP-3968404-B1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES UNIVERSAL DISPLAY CORP (US) 2026-04-01 EP disclosed
US-20260059936-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES UNIVERSAL DISPLAY CORPORATION (US) 2026-02-26 US disclosed
EP-4651875-A2 QUINAZOLINE COMPOUNDS AND USES Prosetta Biosciences, Inc. (US) 2025-11-26 EP disclosed
EP-4010330-B1 QUINOLINE DERIVATIVES AS PROTEIN KINASE INHIBITORS HIRUNDO BIOSCIENCES (BE) 2025-10-01 EP disclosed
US-12390463-B2 Dosage forms and regimens for amino acid compounds PLIANT THERAPEUTICS, INC. (US) 2025-08-19 US disclosed
US-20250223288-A1 AMINO ACID COMPOUNDS AND METHODS OF USE PLIANT THERAPEUTICS, INC. 2025-07-10 US disclosed
EP-4520329-A2 TREATMENT OF RESPIRATORY DISEASES WITH AMINO ACID COMPOUNDS Pliant Therapeutics, Inc. (US) 2025-03-12 EP disclosed
EP-4509512-A2 AMINO ACID COMPOUNDS AND METHODS OF USE Pliant Therapeutics, Inc. (US) 2025-02-19 EP disclosed
US-4808715-A HYPERTENSIVE AGENTS JOHN WYETH & BROTHER LIMITED (GB) 1989-02-28 US disclosed
US-4734510-A HYPOTENSIVE AGENTS JOHN WYETH & BROTHER LIMITED (GB) 1988-03-29 US disclosed
US-4675047-A MONOCOTYLEDON WEES ICI AUSTRALIA LIMITED, 1 NICHOLSON ST., MELBOURNE, VICTORIA, 3000, AUSTRALIA, A CORP. OF AUSTRALIA 1987-06-23 US disclosed
US-4640920-A HYPOTENSIVE AGENTS JOHN WYETH & BROTHER LIMITED (GB) 1987-02-03 US disclosed
US-4464375-A ANALGESIC, ANTIINFLAMMATORY SANKYO CO., LTD. (JP) 1984-08-07 US disclosed
JP-S5913765-A 2-(4-QUINAZOLINYL)AMINOBENZOIC ACID DERIVATIVE KYORIN PHARMACEUT CO LTD 1984-01-24 JP disclosed
US-4322420-A Method of using 4-anilinoquinazoline derivatives as analgesic and anti-inflammatory agents SANKYO COMPANY LIMITED (JP) 1982-03-30 US disclosed
EP-0044163-A2 Quinazolinyloxy(amino)phenoxyalkane carboxylic acid derivatives, process for their synthesis, herbicidal compositions containing them and their use as herbicides ICI AUSTRALIA LIMITED (AU) 1982-01-20 EP disclosed
US-3931179-A ANTIOBESITY SANDOZ INC. (US) 1976-01-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12390463-B2 Dosage forms and regimens for amino acid compounds ITGB6, ITGA6, ITGAV PDE4A 3891/4885PDE4B 3849/4885PDE4C 4382/4885
US-20250223288-A1 AMINO ACID COMPOUNDS AND METHODS OF USE ITGB6, ITGA6, ITGA5 PDE4A 3921/4885PDE4B 3861/4885PDE4C 4299/4885
US-20260059936-A1 ORGANIC ELECTROLUMINESCENT MATERIALS AND DEVICES LBR, GLRB, GLRA1 PDE4A 4879/4885PDE4B 4878/4885PDE4C 4884/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.