SCHEMBL4011663

SCHEMBL4011663

Nc1ncc(-c2cccc(N3CCNCC3)c2)nc1-c1nc2ccccc2[nH]1

nearest known ligand 0.75

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ATR Q13535 16/20 0.75
CDK1 P06493 1/20 0.56
CDK2 P24941 1/20 0.56
MKNK1 Q9BUB5 1/20 0.56
MKNK2 Q9HBH9 1/20 0.56
PRKDC P78527 1/20 0.52
ATM Q13315 1/20 0.52
EGFR P00533 1/20 0.52
PRKCI P41743 1/20 0.50
TGFBR1 P36897 1/20 0.49
ACVR1 Q04771 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4009204 0.92 ATR (0.67) ATRPRKDCATMEGFR
SCHEMBL4016014 0.91 ATR (0.66) ATRPRKDCATMEGFR
SCHEMBL13139379 0.89 ATR (0.70) ATRCDK1CDK2MKNK1MKNK2
SCHEMBL4003249 0.89 ATR (0.64) ATRPRKDCATMEGFR
SCHEMBL4009691 0.89 ATR (0.72) ATRPRKDCATMEGFR
SCHEMBL4009550 0.89 ATR (0.72) ATRPRKDCATMEGFR
SCHEMBL4008991 0.89 ATR (0.60) ATRCDK1CDK2MKNK1MKNK2
SCHEMBL3058004 0.85 ATR (1.00) ATRCDK1CDK2MKNK1MKNK2
SCHEMBL4039257 0.83 ATR (0.80) ATRPRKDCATMEGFR
Hydrochloric Acid SCHEMBL3511276 0.81 HTR7 (0.57) ATR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007390-A2 2-PYRAZ INYLBENZ IMIDAZOLE DERIVATIVES AS RECEPTOR TYROSINE KINASE INHIBITORS ASTRAZENECA AB (SE) 2009-01-15 WO claimed
WO-2009007390-A2 2-PYRAZ INYLBENZ IMIDAZOLE DERIVATIVES AS RECEPTOR TYROSINE KINASE INHIBITORS ASTRAZENECA AB (SE) 2009-01-15 WO disclosed