SCHEMBL4011960

SCHEMBL4011960

Nc1cc(-c2cccc(Br)c2)c2cccc(C(F)(F)F)c2n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.41
BACE1 P56817 2/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
NR1H2 P55055 6/20 0.40
NR1H3 Q13133 6/20 0.40
KDM4E B2RXH2 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
ALDH1A1 P00352 2/20 0.38
MAPT P10636 2/20 0.38
HPGD P15428 2/20 0.38
RAB9A P51151 2/20 0.38
NPC1 O15118 1/20 0.38
POLB P06746 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
HSD17B10 Q99714 1/20 0.38
HK1 P19367 1/20 0.38
HKDC1 Q2TB90 1/20 0.38
RXRA P19793 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4012984 0.78 NR1H2 (0.62) MEN1KMT2ANR1H2NR1H3RXRA
SCHEMBL4011578 0.78 NR1H2 (0.69) NR1H2NR1H3RXRA
SCHEMBL3508106 0.75 ESR1 (0.42) ESR1MEN1KMT2ANR1H2NR1H3
SCHEMBL3507631 0.75 ESR1 (0.42) ESR1MEN1KMT2ANR1H2ALDH1A1
SCHEMBL31690946 0.74 BACE1 (0.50) ESR1BACE1KMT2ANR1H2NR1H3
SCHEMBL4018001 0.73 KDM4E (0.51) ESR1MEN1KMT2ANR1H2NR1H3
SCHEMBL31690861 0.73 BACE1 (0.49) ESR1BACE1KMT2ANR1H2NR1H3
SCHEMBL3507644 0.73 ESR1 (0.46) ESR1MEN1KMT2ANR1H2NR1H3
SCHEMBL4012785 0.72 NR1H2 (0.42) ESR1NR1H2NR1H3IKBKBAURKA
SCHEMBL4012404 0.72 ESR1 (0.44) ESR1NR1H2NR1H3RXFP1IKBKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101541751-A Quinoline compounds WYETH CORP (US) 2009-09-23 CN disclosed
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed