SCHEMBL4011978

SCHEMBL4011978

O=S1(=O)CCc2ccc(F)cc21

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.54
CA2 P00918 3/20 0.54
CA9 Q16790 2/20 0.54
PTGDR2 Q9Y5Y4 4/20 0.44
PARP1 P09874 1/20 0.37
PARP10 Q53GL7 1/20 0.37
CA12 O43570 1/20 0.36
CA4 P22748 1/20 0.36
CA7 P43166 1/20 0.36
LMNA P02545 1/20 0.35
KDM4E B2RXH2 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
GRIA2 P42262 2/20 0.34
GRIA1 P42261 1/20 0.34
GRIA3 P42263 1/20 0.34
GRIA4 P48058 1/20 0.34
VEGFA P15692 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13547786 0.76 CA1 (0.54) CA1CA2CA9PTGDR2PARP1
SCHEMBL30635417 0.76 CA2 (0.54) CA1CA2CA9PTGDR2PARP1
SCHEMBL1155659 0.76 CA9 (0.59) CA1CA2CA9PTGDR2CA12
SCHEMBL10444145 0.76 CA2 (0.54) CA1CA2CA9PTGDR2PARP1
SCHEMBL24141272 0.76 CA1 (0.50) CA1CA2CA9PTGDR2PARP1
SCHEMBL7873031 0.76 CA2 (0.37) CA1CA2CA9PARP1PARP10
SCHEMBL21028030 0.73 CA2 (0.51) CA1CA2CA9PTGDR2KDM4E
SCHEMBL10199637 0.72 CA1 (0.50) CA1CA2CA9
SCHEMBL10443651 0.72 CA9 (0.50) CA1CA2CA9PTGDR2CA12
SCHEMBL14456114 0.72 CA1 (0.50) CA1CA2CA9PTGDR2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed