SCHEMBL4012011

SCHEMBL4012011

Cc1cc(-c2cc(OCc3cccc(S(C)(=O)=O)c3)ccc2F)c2cccc(C(F)(F)F)c2n1

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NR1H3 Q13133 15/20 0.47
NR1H2 P55055 14/20 0.47
RXRA P19793 1/20 0.45
CYP4F2 P78329 1/20 0.42
CYP4A11 Q02928 1/20 0.42
PTK2 Q05397 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4014198 0.90 NR1H3 (0.47) NR1H3NR1H2RXRACYP4F2CYP4A11
SCHEMBL4014463 0.88 NR1H2 (0.43) NR1H3NR1H2CYP4F2CYP4A11
SCHEMBL4010727 0.87 NR1H3 (0.58) NR1H3NR1H2RXRA
SCHEMBL4012268 0.86 NR1H2 (0.58) NR1H3NR1H2RXRA
SCHEMBL3507031 0.83 NR1H3 (0.46) NR1H3NR1H2RXRACYP4F2CYP4A11
SCHEMBL4012475 0.81 NR1H2 (0.58) NR1H3NR1H2RXRA
SCHEMBL4014419 0.80 NR1H2 (0.56) NR1H3NR1H2RXRA
SCHEMBL4012195 0.80 NR1H2 (0.45) NR1H3NR1H2CYP4F2CYP4A11
SCHEMBL3507588 0.79 NR1H3 (0.46) NR1H3NR1H2RXRACYP4F2CYP4A11
SCHEMBL4014835 0.79 NR1H2 (0.39) NR1H3NR1H2RXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP claimed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO claimed
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed