SCHEMBL4012749

SCHEMBL4012749

CCCc1nc(CC)c(CC(C)CO)c(=O)n1Cc1ccc(-c2ccccc2-c2noc(=O)[nH]2)cc1

nearest known ligand 0.64

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 6/20 0.64
PPARG P37231 14/20 0.62
KCNH2 Q12809 2/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1894931 0.85 AGTR1 (0.60) AGTR1PPARGKCNH2
SCHEMBL1897713 0.84 SLC33A1 (0.61) AGTR1PPARG
SCHEMBL1893484 0.83 AGTR1 (0.63) AGTR1PPARGKCNH2
SCHEMBL4011284 0.83 PPARG (0.56) AGTR1PPARG
SCHEMBL1895203 0.82 PPARG (0.57) AGTR1PPARGKCNH2
SCHEMBL12348495 0.81 PPARG (0.60) AGTR1PPARG
SCHEMBL1892292 0.81 PPARG (0.56) AGTR1PPARGKCNH2
SCHEMBL1887274 0.81 AGTR1 (0.59) AGTR1PPARGKCNH2
SCHEMBL1893527 0.81 AGTR1 (0.59) AGTR1PPARGKCNH2
SCHEMBL1890877 0.80 PPARG (0.54) AGTR1PPARGKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009133970-A1 CRYSTALLINE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-11-05 WO disclosed
EP-2074117-A2 HETEROMONOCYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2009-07-01 EP disclosed
WO-2008062905-A2 HETEROMONOCYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-05-29 WO disclosed