SCHEMBL4012804

SCHEMBL4012804

CCCCC1=C(Cc2ccc(-c3ccccc3-c3noc(=O)[nH]3)cc2)CN(c2ccc(OCC)cc2)C(C)=N1

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SLC33A1 O00400 6/20 0.47
PPARG P37231 7/20 0.45
AGTR1 P30556 2/20 0.45
ALDH1A1 P00352 1/20 0.44
LTB4R2 Q9NPC1 1/20 0.44
KCNH2 Q12809 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4011144 0.93 SLC33A1 (0.47) SLC33A1PPARGAGTR1
SCHEMBL4010722 0.91 PPARG (0.45) SLC33A1PPARGAGTR1
SCHEMBL4016064 0.90 SLC33A1 (0.48) SLC33A1PPARG
SCHEMBL4016688 0.88 PPARG (0.47) PPARGAGTR1
SCHEMBL4312498 0.87 PPARG (0.45) SLC33A1PPARGAGTR1
SCHEMBL4017556 0.87 PPARG (0.45) SLC33A1PPARGAGTR1
SCHEMBL4016515 0.86 SLC33A1 (0.47) SLC33A1PPARGAGTR1
SCHEMBL4013359 0.86 SLC33A1 (0.47) SLC33A1PPARGAGTR1
SCHEMBL4010901 0.85 PPARG (0.44) SLC33A1PPARGAGTR1
SCHEMBL4010601 0.84 AGTR1 (0.45) SLC33A1PPARGAGTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009133970-A1 CRYSTALLINE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-11-05 WO disclosed
EP-2074117-A2 HETEROMONOCYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2009-07-01 EP disclosed
WO-2008062905-A2 HETEROMONOCYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-05-29 WO disclosed