SCHEMBL4013268

SCHEMBL4013268

NS(=O)(=O)c1cccc(-c2cccc(-c3ccnc4c(C(F)(F)F)cccc34)c2)c1

nearest known ligand 0.81

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 15/20 0.81
NR1H3 Q13133 14/20 0.81
RXRA P19793 1/20 0.64
IKBKB O14920 1/20 0.53
CHUK O15111 1/20 0.53
CA12 O43570 2/20 0.48
CA1 P00915 2/20 0.48
CA2 P00918 2/20 0.48
CA9 Q16790 2/20 0.48
SYK P43405 1/20 0.48
PPARG P37231 1/20 0.46
LRRK2 Q5S007 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4012168 0.89 NR1H2 (1.00) NR1H2NR1H3RXRA
SCHEMBL4010294 0.87 NR1H2 (1.00) NR1H2NR1H3RXRAPPARG
SCHEMBL4013652 0.87 NR1H2 (0.95) NR1H2NR1H3RXRA
SCHEMBL4014617 0.86 NR1H2 (0.78) NR1H2NR1H3RXRASYKPPARG
SCHEMBL4012992 0.86 NR1H2 (0.79) NR1H2NR1H3RXRAPPARG
SCHEMBL4018359 0.84 NR1H2 (0.86) NR1H2NR1H3RXRAPPARG
SCHEMBL4013224 0.84 NR1H2 (0.77) NR1H2NR1H3RXRAPPARG
SCHEMBL4012032 0.84 NR1H2 (0.85) NR1H2NR1H3RXRASYK
SCHEMBL4009753 0.84 NR1H2 (0.73) NR1H2NR1H3RXRAPPARG
SCHEMBL4013299 0.84 NR1H2 (0.77) NR1H2NR1H3RXRAPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP claimed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO claimed