SCHEMBL4013350

SCHEMBL4013350

COc1cc(-c2cnc(N)c(C(=O)O)n2)ccc1O

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NEK2 P51955 6/20 0.58
FYN P06241 8/20 0.53
CHEK2 O96017 3/20 0.52
CHEK1 O14757 1/20 0.52
TGFBR1 P36897 1/20 0.50
PIK3CD O00329 1/20 0.49
PIK3CA P42336 1/20 0.49
PIK3CG P48736 1/20 0.49
PRKDC P78527 1/20 0.48
ATR Q13535 1/20 0.48
ALDH1A1 P00352 1/20 0.48
GAA P10253 1/20 0.48
ALOX15 P16050 1/20 0.48
HSD17B10 Q99714 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4008712 0.85 FYN (0.51) NEK2FYNPIK3CAALDH1A1GAA
SCHEMBL11907493 0.83 NEK2 (0.72) NEK2FYN
SCHEMBL23703221 0.81 ATR (0.48) NEK2PIK3CDPIK3CAPIK3CGPRKDC
SCHEMBL11907360 0.80 ATR (0.70) NEK2CHEK1PRKDCATR
SCHEMBL4011105 0.77 MCHR1 (0.52) NEK2ATR
SCHEMBL11908281 0.77 ATR (0.67) PIK3CGPRKDCATR
SCHEMBL3461060 0.77 PIK3CD (0.67) NEK2PIK3CDPIK3CAPIK3CGPRKDC
SCHEMBL11909602 0.76 MAP4K4 (0.50) NEK2PRKDCATR
SCHEMBL30048631 0.76 ATR (0.67) PRKDCATR
SCHEMBL23703073 0.76 ATR (0.67) PRKDCATR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007390-A2 2-PYRAZ INYLBENZ IMIDAZOLE DERIVATIVES AS RECEPTOR TYROSINE KINASE INHIBITORS ASTRAZENECA AB (SE) 2009-01-15 WO disclosed