SCHEMBL4011105

SCHEMBL4011105

COc1cc(-c2cnc(N)c(C(=O)O)n2)ccc1OCCN1CCCC1

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 10/20 0.52
NEK2 P51955 3/20 0.51
CCNE2 O96020 1/20 0.49
CCNE1 P24864 1/20 0.49
CDK2 P24941 1/20 0.49
GSK3B P49841 1/20 0.49
MAP3K11 Q16584 1/20 0.48
ADORA2A P29274 2/20 0.48
ADORA1 P30542 1/20 0.48
LTA4H P09960 1/20 0.47
HRH3 Q9Y5N1 1/20 0.47
ATR Q13535 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3936085 0.81 NEK2 (0.47) NEK2MAP3K11ATR
SCHEMBL4013350 0.77 NEK2 (0.58) NEK2ATR
SCHEMBL220877 0.77 NOS3 (0.61) MCHR1ADORA2AADORA1LTA4HHRH3
SCHEMBL3928126 0.76 MCHR1 (0.47) MCHR1MAP3K11ADORA2AADORA1LTA4H
SCHEMBL4008321 0.76 ATR (0.55) MCHR1MAP3K11ADORA2AADORA1ATR
SCHEMBL15333931 0.76 LTA4H (0.49) MCHR1ADORA2AADORA1LTA4H
SCHEMBL4006573 0.75 ATR (0.59) ATR
SCHEMBL4012928 0.75 ATR (0.54) MCHR1CDK2MAP3K11ADORA2AADORA1
Hydrochloric Acid SCHEMBL7427266 0.74 MCHR1 (0.53) MCHR1ADORA2AADORA1HRH3
SCHEMBL15333915 0.74 FYN (0.56) MCHR1ADORA2AADORA1LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007390-A2 2-PYRAZ INYLBENZ IMIDAZOLE DERIVATIVES AS RECEPTOR TYROSINE KINASE INHIBITORS ASTRAZENECA AB (SE) 2009-01-15 WO disclosed