SCHEMBL4014149

SCHEMBL4014149

Cc1cc(N(C)c2nccc(Nc3cc(CCc4cccc(C(=O)N(C)C)c4)[nH]n3)n2)on1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 12/20 0.51
IGF1R P08069 12/20 0.51
KDR P35968 11/20 0.51
INSR P06213 2/20 0.45
ALDH1A1 P00352 2/20 0.38
CYP1A2 P05177 2/20 0.38
CYP3A4 P08684 2/20 0.38
MAPK1 P28482 2/20 0.38
HPGD P15428 1/20 0.38
TSHR P16473 1/20 0.38
CYP2C19 P33261 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
EPHB4 P54760 1/20 0.36
AURKA O14965 1/20 0.35
PAK1 Q13153 1/20 0.35
USP2 O75604 1/20 0.35
CYP2D6 P10635 1/20 0.35
EGFR P00533 1/20 0.34
BRD4 O60885 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4014156 0.84 IGF1R (0.73) FGFR1IGF1RKDRINSR
SCHEMBL4013739 0.84 FGFR1 (0.52) FGFR1IGF1RKDRINSRALDH1A1
SCHEMBL4007933 0.81 FGFR1 (0.37) FGFR1IGF1RKDRINSRALDH1A1
Hydrochloric Acid SCHEMBL4009909 0.81 FGFR1 (0.48) FGFR1IGF1RKDRINSRAURKA
SCHEMBL5103524 0.78 FGFR1 (0.56) FGFR1IGF1RKDRINSRAURKA
SCHEMBL5096876 0.77 FGFR1 (0.40) FGFR1IGF1RKDRINSR
SCHEMBL5100451 0.74 MRGPRX4 (0.38) SMN1; SMN2
SCHEMBL5096788 0.73 IGF1R (0.34) FGFR1IGF1RKDRINSRALDH1A1
Hydrochloric Acid SCHEMBL5110836 0.73 MRGPRX4 (0.37) SMN1; SMN2
SCHEMBL4012455 0.73 FGFR1 (0.48) FGFR1IGF1RKDRINSRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2044063-A1 PYRIMIDINE DERIVATIVES USEFUL IN THE TREATMENT OF CANCER Astra Zeneca AB (SE) 2009-04-08 EP disclosed
WO-2008001070-A1 PYRIMIDINE DERIVATIVES USEFUL IN THE TREATMENT OF CANCER ASTRAZENECA AB (SE) 2008-01-03 WO disclosed
US-20080004302-A1 Novel Compounds ASTRAZENECA AB (SE) 2008-01-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080004302-A1 Novel Compounds CYP11B2, CYP11B1, CYP46A1 FGFR1 1428/4885IGF1R 3217/4885KDR 3815/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.