SCHEMBL4015590

SCHEMBL4015590

Cc1ccc(Cl)c(CC#N)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 2/20 0.39
GABRG2 P18507 2/20 0.39
GABRB3 P28472 2/20 0.39
GABRB2 P47870 1/20 0.39
SLC6A4 P31645 2/20 0.38
HTR2A P28223 1/20 0.38
KCNH2 Q12809 1/20 0.38
CYP2A6 P11509 1/20 0.38
CSNK2A1 P68400 1/20 0.36
HPGD P15428 2/20 0.35
ALDH1A1 P00352 2/20 0.35
MEN1 O00255 1/20 0.35
USP2 O75604 1/20 0.35
POLB P06746 1/20 0.35
MAPT P10636 1/20 0.35
CYP2C9 P11712 1/20 0.35
ALOX12 P18054 1/20 0.35
MAPK1 P28482 1/20 0.35
CYP2C19 P33261 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2581205 0.79 CYP2A6 (0.51) GABRA1GABRG2GABRB3GABRB2SLC6A4
Water SCHEMBL17670054 0.79 TAAR1 (0.50) HPGDALDH1A1MEN1POLBMAPT
SCHEMBL1019451 0.79 TAAR1 (0.50) HPGDALDH1A1MEN1POLBMAPT
SCHEMBL30453664 0.79 CYP2A6 (0.51) GABRA1GABRG2GABRB3GABRB2SLC6A4
SCHEMBL24786214 0.76 AR (0.41) CYP2A6ALDH1A1GAAFFAR1
SCHEMBL3067521 0.76 AMY1A (0.53) CSNK2A1HPGDALDH1A1MEN1MAPT
SCHEMBL155058 0.76 CSNK2A1 (0.49) SLC6A4HTR2AKCNH2CYP2A6CSNK2A1
SCHEMBL5642630 0.76 KCNH2 (0.39) SLC6A4HTR2AKCNH2CYP2A6CSNK2A1
SCHEMBL952178 0.76 TAAR1 (0.38) SLC6A4CYP2A6ALDH1A1MAPK1TAAR1
SCHEMBL6036428 0.76 TAAR1 (0.34) KCNH2CYP2A6CSNK2A1HPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3943087-A1 HETEROARYL COMPOUNDS AND USES THEREOF Celgene CAR LLC (BM) 2022-01-26 EP disclosed
WO-2009085797-A1 PROCESSES FOR PREPARING HIV REVERSE TRANSCRIPTASE INHIBITORS GILEAD SCIENCES, INC. (US) 2009-07-09 WO disclosed
US-3944571-A ANTIARTHRITIC SMITHKLINE CORPORATION (US) 1976-03-16 US disclosed