SCHEMBL4015645

SCHEMBL4015645

CCCc1nc(=O)c(Oc2ccc(OC)cc2)c(C)n1Cc1ccc(-c2ccccc2C#N)cc1

nearest known ligand 0.57

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PPARG P37231 6/20 0.57
NPBWR1 P48145 1/20 0.45
AGTR1 P30556 3/20 0.42
AGTR2 P50052 2/20 0.42
MAPT P10636 1/20 0.42
MAPK1 P28482 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
ACHE P22303 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4016128 0.94 PPARG (0.60) PPARGAGTR1ACHE
SCHEMBL1891952 0.90 PPARG (0.57) PPARGNPBWR1AGTR1AGTR2MAPT
SCHEMBL4012577 0.86 PPARG (0.57) PPARGAGTR1AGTR2ACHE
SCHEMBL4016070 0.84 PPARG (0.57) PPARGAGTR1AGTR2MAPTMAPK1
SCHEMBL4007590 0.84 PPARG (0.53) PPARGAGTR1ACHE
SCHEMBL1898235 0.83 PPARG (0.60) PPARGAGTR1ACHE
SCHEMBL4009893 0.83 PPARG (0.51) PPARGAGTR1AGTR2
SCHEMBL4012027 0.82 PPARG (0.63) PPARGAGTR1AGTR2MAPK1ACHE
SCHEMBL1892312 0.81 PPARG (0.58) PPARGAGTR1MAPTMAPK1NPSR1
SCHEMBL1893323 0.81 PPARG (0.58) PPARGAGTR1AGTR2ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009133970-A1 CRYSTALLINE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-11-05 WO disclosed
EP-2074117-A2 HETEROMONOCYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2009-07-01 EP disclosed
WO-2008062905-A2 HETEROMONOCYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-05-29 WO disclosed