SCHEMBL4016424

SCHEMBL4016424

CC(C)C(O)C(=O)NCC1CCN(C(=O)OC(C)(C)C)CC1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.57
PKM P14618 1/20 0.57
KMT2A Q03164 1/20 0.44
EPHX1 P07099 1/20 0.44
NPC1 O15118 1/20 0.44
ALDH1A1 P00352 1/20 0.44
MAPT P10636 1/20 0.44
MAPK1 P28482 1/20 0.44
HTT P42858 1/20 0.44
RAB9A P51151 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
GPR119 Q8TDV5 5/20 0.43
FPR3 P25089 1/20 0.43
FPR2 P25090 1/20 0.43
HPGD P15428 1/20 0.43
TGFBR1 P36897 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
RECQL P46063 1/20 0.41
KEAP1 Q14145 1/20 0.41
NFE2L2 Q16236 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4016421 1.00 KDM4E (0.57) KDM4EPKMKMT2AEPHX1NPC1
SCHEMBL19652088 0.88 KDM4E (0.60) KDM4EPKMKMT2AEPHX1NPC1
SCHEMBL21176252 0.88 KDM4E (0.53) KDM4EPKMKMT2AEPHX1NPC1
SCHEMBL21176375 0.85 KDM4E (0.50) KDM4EPKMKMT2AEPHX1NPC1
SCHEMBL21176196 0.81 KDM4E (0.47) KDM4EPKMKMT2AEPHX1NPC1
SCHEMBL21176301 0.81 KDM4E (0.48) KDM4EPKMKMT2AEPHX1GPR119
SCHEMBL24853346 0.81 KDM4E (0.64) KDM4EPKMEPHX1FPR3FPR2
SCHEMBL1245476 0.81 KDM4E (0.64) KDM4EPKMEPHX1GPR119FPR3
SCHEMBL6152939 0.81 KDM4E (0.68) KDM4EPKMEPHX1GPR119FPR3
SCHEMBL28767036 0.81 EPHX2 (0.40) KDM4EPKMKMT2AEPHX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1784393-B1 QUINAZOLINES USEFUL AS MODULATORS OF ION CHANNELS VERTEX PHARMA (US) 2009-07-01 EP disclosed