SCHEMBL4017280

SCHEMBL4017280

CCS(=O)(=O)c1cccc(Oc2cccc(-c3ccnc4c(C#N)cccc34)c2)c1

nearest known ligand 0.58

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 18/20 0.58
NR1H3 Q13133 18/20 0.58
RXRA P19793 1/20 0.56
LRRK2 Q5S007 1/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4016986 0.93 NR1H2 (0.56) NR1H2NR1H3RXRALRRK2PTGDR2
SCHEMBL4016541 0.93 NR1H2 (0.52) NR1H2NR1H3RXRALRRK2PTGDR2
SCHEMBL4012434 0.91 NR1H2 (0.52) NR1H2NR1H3RXRALRRK2PTGDR2
SCHEMBL4011793 0.90 NR1H2 (0.72) NR1H2NR1H3RXRA
SCHEMBL4013990 0.89 NR1H2 (0.52) NR1H2NR1H3RXRAPTGDR2
SCHEMBL4017885 0.88 NR1H2 (0.52) NR1H2NR1H3RXRAPTGDR2
SCHEMBL4017312 0.87 NR1H2 (0.71) NR1H2NR1H3RXRALRRK2PTGDR2
SCHEMBL4012271 0.85 NR1H2 (0.62) NR1H2NR1H3RXRA
SCHEMBL4015112 0.85 NR1H2 (0.62) NR1H2NR1H3RXRALRRK2
SCHEMBL4013225 0.85 NR1H2 (0.80) NR1H2NR1H3RXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP claimed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO claimed
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed