SCHEMBL4017757

SCHEMBL4017757

CCCc1nc(=O)c(-c2ccc(O)cc2)c(C)n1Cc1ccc(-c2ccccc2C#N)cc1

nearest known ligand 0.60

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PPARG P37231 8/20 0.60
ESR2 Q92731 1/20 0.44
ACHE P22303 1/20 0.43
ALDH1A1 P00352 1/20 0.43
MAPK1 P28482 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4012027 0.93 PPARG (0.63) PPARGACHEALDH1A1MAPK1
SCHEMBL4012581 0.90 PPARG (0.59) PPARGESR2ACHE
SCHEMBL1890122 0.88 PPARG (0.61) PPARGESR2ACHE
SCHEMBL4010868 0.87 PPARG (0.55) PPARGACHEALDH1A1MAPK1
SCHEMBL4009715 0.85 PPARG (0.53) PPARGACHE
SCHEMBL1892413 0.85 PPARG (0.60) PPARGESR2
SCHEMBL4017163 0.83 PPARG (0.62) PPARGACHE
SCHEMBL12737302 0.82 PPARG (0.71) PPARGACHE
SCHEMBL4014913 0.82 PPARG (0.49) PPARGACHE
SCHEMBL4016128 0.81 PPARG (0.60) PPARGACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009133970-A1 CRYSTALLINE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-11-05 WO disclosed
EP-2074117-A2 HETEROMONOCYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2009-07-01 EP disclosed
WO-2008062905-A2 HETEROMONOCYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-05-29 WO disclosed