SCHEMBL4020356

SCHEMBL4020356

Cc1nc(C2CCC(C(C)C)CC2)c(-c2ccc(Cl)cc2)c(=O)[nH]1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 3/20 0.41
TYMS P04818 2/20 0.39
PSD A5PKW4 4/20 0.36
CNR1 P21554 1/20 0.35
GABRA1 P14867 1/20 0.34
GABRG2 P18507 1/20 0.34
GABRB3 P28472 1/20 0.34
PDE2A O00408 4/20 0.34
MAPK1 P28482 1/20 0.34
MDM2 Q00987 1/20 0.33
SLC2A1 P11166 1/20 0.33
CSF1R P07333 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4020354 1.00 TRPV1 (0.41) TRPV1TYMSPSDCNR1GABRA1
SCHEMBL13747129 0.82 TYMS (0.38) TRPV1TYMSPSDCNR1GABRA1
SCHEMBL13746236 0.80 TYMS (0.41) TRPV1TYMSPSDCNR1GABRA1
SCHEMBL13746305 0.80 TYMS (0.41) TRPV1TYMSPSDCNR1GABRA1
SCHEMBL13746410 0.76 TYMS (0.39) TRPV1TYMSPSDCNR1PDE2A
SCHEMBL13746006 0.76 TYMS (0.39) TRPV1TYMSPSDCNR1GABRA1
SCHEMBL13746092 0.74 PSD (0.38) TRPV1TYMSPSDCNR1GABRA1
SCHEMBL4192359 0.74 PSD (0.38) TRPV1TYMSPSDCNR1GABRA1
SCHEMBL13746104 0.73 TYMS (0.38) TRPV1TYMSPSDCNR1PDE2A
SCHEMBL13746667 0.70 PDE2A (0.37) TYMSPDE2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009100403-A1 SUBSTITUTED ARYL PYRIMIDINONES NEUROGEN CORPORATION (US) 2009-08-13 WO disclosed