SCHEMBL4021070

SCHEMBL4021070

FC(F)(F)c1cc(COC[C@@H]2NCCN(Cc3ccccc3)[C@@H]2c2ccccc2)cc(C(F)(F)F)c1

nearest known ligand 0.58

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 19/20 0.58
TP53 P04637 2/20 0.45
CYP1A2 P05177 2/20 0.45
CYP3A4 P08684 2/20 0.45
CYP2D6 P10635 2/20 0.45
TSHR P16473 2/20 0.45
TACR2 P21452 1/20 0.45
TACR3 P29371 1/20 0.45
MEN1 O00255 1/20 0.45
MAPT P10636 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
KMT2A Q03164 1/20 0.45
THPO P40225 1/20 0.45
HSD17B10 Q99714 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4023056 0.99 TACR1 (0.57) TACR1TP53CYP1A2CYP3A4CYP2D6
SCHEMBL4027731 0.86 TACR1 (0.66) TACR1CYP3A4TACR2TACR3
Hydrochloric Acid SCHEMBL4021098 0.85 TACR1 (0.65) TACR1CYP3A4TACR2TACR3
SCHEMBL4024411 0.82 TACR1 (0.52) TACR1TACR2TACR3
SCHEMBL4027291 0.78 TACR1 (0.62) TACR1TP53CYP1A2CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL4028643 0.77 MEN1 (0.61) TACR1TP53CYP1A2CYP3A4CYP2D6
SCHEMBL9024514 0.74 TACR1 (1.00) TACR1
SCHEMBL9366823 0.74 TACR1 (1.00) TACR1
SCHEMBL264225 0.73 TACR1 (0.76) TACR1TACR2TACR3
SCHEMBL7022339 0.73 TACR1 (0.76) TACR1TACR2TACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1338592-B1 Novel 2-phenylpiperazine derivatives NIPPON ZOKI PHARMACEUTICAL CO (JP) 2009-01-21 EP claimed