SCHEMBL4021172

SCHEMBL4021172

COc1ccc2c(c1)c(CC(=O)OCCCCO[N+](=O)[O-])c(C)n2C(=O)c1ccc(Cl)cc1

nearest known ligand 0.79

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 17/20 0.79
PTGS1 P23219 5/20 0.77
CNR2 P34972 1/20 0.69
AKR1C3 P42330 1/20 0.69
HTR1A P08908 1/20 0.69
PKM P14618 1/20 0.69
GLO1 Q04760 1/20 0.69
HIF1A Q16665 1/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12106520 0.91 PTGS2 (0.71) PTGS2PTGS1CNR2AKR1C3HTR1A
SCHEMBL6754016 0.88 PTGS2 (0.88) PTGS2PTGS1CNR2AKR1C3HTR1A
SCHEMBL220697 0.87 PTGS2 (0.78) PTGS2PTGS1CNR2AKR1C3HTR1A
SCHEMBL29170168 0.87 PTGS2 (0.86) PTGS2PTGS1CNR2AKR1C3HTR1A
SCHEMBL5806528 0.87 PTGS2 (1.00) PTGS2PTGS1
SCHEMBL217602 0.86 PTGS2 (0.68) PTGS2PTGS1CNR2AKR1C3HTR1A
SCHEMBL16010166 0.86 PTGS2 (0.84) PTGS2PTGS1CNR2AKR1C3HTR1A
SCHEMBL12742120 0.86 PTGS2 (0.91) PTGS2PTGS1CNR2AKR1C3HTR1A
SCHEMBL30077218 0.86 PTGS2 (0.91) PTGS2PTGS1CNR2AKR1C3HTR1A
SCHEMBL13813542 0.86 PTGS2 (1.00) PTGS2PTGS1CNR2AKR1C3HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1154999-B1 NITROXYDERIVATIVES HAVING ANTIINFLAMMATORY, ANALGESIC AND ANTITHROMBOTIC ACTIVITY NICOX SA (FR) 2009-04-15 EP disclosed
US-6613784-B1 Cyclooxygenase inhibitors such as 2-acetyloxybenzoic acid 6-(nitroxymethyl)-2-methylpyridinyl ester hydrochloride, having good kinetics, solubility and efficiency; nontoxic NICOX S.A. (FR) 2003-09-02 US disclosed
CN-1342147-A Nitrooxyderivatives having anti-inflammatory, analgesic and antithrombotic activity NICOX SA (FR) 2002-03-27 CN disclosed
EP-1154999-A1 NITROXYDERIVATIVES HAVING ANTIINFLAMMATORY, ANALGESIC AND ANTITHROMBOTIC ACTIVITY NICOX S.A. (FR) 2001-11-21 EP disclosed
WO-2000051988-A1 NITROXYDERIVATIVES HAVING ANTIINFLAMMATORY, ANALGESIC AND ANTITHROMBOTIC ACTIVITY NICOX S.A. (FR) 2000-09-08 WO disclosed