SCHEMBL4021802

SCHEMBL4021802

COc1cc(N2CCN(C(C=O)n3nc(CC(C)O)c(Cl)c3C)CC2)c(F)cc1F

nearest known ligand 0.35

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 16/20 0.35
FFAR4 Q5NUL3 1/20 0.34
CYP2C19 P33261 1/20 0.32
KCNH2 Q12809 1/20 0.32
MAPT P10636 1/20 0.31
NPM1 P06748 1/20 0.31
ALK Q9UM73 1/20 0.31
JAK2 O60674 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4453143 0.82 CCR1 (0.51) CCR1CYP2C19KCNH2
SCHEMBL4016337 0.78 CCR1 (0.37) CCR1CYP2C19KCNH2MAPT
SCHEMBL4018792 0.77 CCR1 (0.47) CCR1CYP2C19KCNH2
SCHEMBL4019585 0.76 CCR1 (0.43) CCR1CYP2C19KCNH2MAPT
SCHEMBL4021523 0.76 CCR1 (0.43) CCR1CYP2C19KCNH2MAPT
SCHEMBL3866250 0.75 ALDH1A1 (0.35) CCR1CYP2C19KCNH2MAPTALK
SCHEMBL4311232 0.73 CCR1 (0.61) CCR1CYP2C19KCNH2
SCHEMBL4565941 0.71 CCR1 (0.55) CCR1CYP2C19KCNH2
SCHEMBL4019909 0.71 CCR1 (0.54) CCR1CYP2C19KCNH2
SCHEMBL4019367 0.71 CCR1 (0.49) CCR1CYP2C19KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1691810-A4 SUBSTITUTED PIPERAZINES CHEMOCENTRYX INC (US) 2009-07-01 EP disclosed
EP-1691810-A1 SUBSTITUTED PIPERAZINES ChemoCentryx Inc (US) 2006-08-23 EP disclosed
WO-2005056015-A1 SUBSTITUTED PIPERAZINES CHEMOCENTRYX, INC. (US) 2005-06-23 WO disclosed