SCHEMBL4023670

SCHEMBL4023670

NC(N)=NCc1ccccc1Cl

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 4/20 0.73
HTR3E A5X5Y0 3/20 0.67
HTR3B O95264 3/20 0.67
HTR3A P46098 3/20 0.67
HTR3D Q70Z44 3/20 0.67
HTR3C Q8WXA8 3/20 0.67
GRIN2B Q13224 4/20 0.58
GRIN1 Q05586 3/20 0.58
PKM P14618 1/20 0.52
PNMT P11086 1/20 0.50
IDO1 P14902 4/20 0.47
LMNA P02545 2/20 0.47
HTT P42858 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
HRH4 Q9H3N8 3/20 0.47
HRH3 Q9Y5N1 2/20 0.47
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5068041 0.86 TAAR1 (0.66) TAAR1HTR3EHTR3BHTR3AHTR3D
Hydrochloric Acid SCHEMBL4797248 0.84 TAAR1 (0.64) TAAR1HTR3EHTR3BHTR3AHTR3D
SCHEMBL11588057 0.81 TAAR1 (0.59) TAAR1HTR3EHTR3BHTR3AHTR3D
SCHEMBL9474594 0.76 TAAR1 (0.54) TAAR1HTR3EHTR3BHTR3AHTR3D
SCHEMBL3817964 0.75 CYP1A2 (0.47) TAAR1HTR3EHTR3BHTR3AHTR3D
SCHEMBL7979449 0.73 GRIN2B (1.00) TAAR1HTR3EHTR3BHTR3AHTR3D
SCHEMBL7762998 0.73 GRIN2B (0.54) TAAR1HTR3EHTR3BHTR3AHTR3D
SCHEMBL7763001 0.73 GRIN2B (0.54) TAAR1HTR3EHTR3BHTR3AHTR3D
SCHEMBL2995781 0.73 IDO1 (0.52) TAAR1HTR3EHTR3BHTR3AHTR3D
Hydrochloric Acid SCHEMBL4741263 0.72 TAAR1 (0.50) TAAR1HTR3EHTR3BHTR3AHTR3D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1917244-A2 HETARYL-SUBSTITUTED GUANIDINE COMPOUNDS AND USE THEREOF AS BINDING PARTNERS FOR 5-HT5-RECEPTORS Abbott GmbH & Co. KG (DE) 2008-05-07 EP claimed
WO-2007022964-A2 HETARYL-SUBSTITUTED GUANIDINE COMPOUNDS AND USE THEREOF AS BINDING PARTNERS FOR 5-HT5-RECEPTORS ABBOTT GMBH & CO. KG (DE) 2007-03-01 WO claimed
WO-2009087395-A1 WEIGHT REDUCING COMPOUNDS UNIVERSITY OF STRATHCLYDE (GB) 2009-07-16 WO disclosed