SCHEMBL4023743

SCHEMBL4023743

CCNC(=O)c1ccc2cc(C(O)(c3c[nH]cn3)C(C)C)ccc2c1

nearest known ligand 0.67

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 16/20 0.67
CYP3A4 P08684 14/20 0.67
HPGDS O60760 1/20 0.39
ACSS2 Q9NR19 1/20 0.38
RIPK1 Q13546 1/20 0.38
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4024213 1.00 CYP17A1 (0.67) CYP17A1CYP3A4HPGDSACSS2RIPK1
SCHEMBL4026880 0.90 CYP17A1 (0.60) CYP17A1CYP3A4
SCHEMBL4028778 0.90 CYP17A1 (0.54) CYP17A1CYP3A4
SCHEMBL4027776 0.90 CYP17A1 (0.57) CYP17A1CYP3A4ACSS2
SCHEMBL7533841 0.88 CYP17A1 (0.53) CYP17A1CYP3A4
SCHEMBL4025340 0.88 CYP17A1 (0.65) CYP17A1CYP3A4CYP2C9CYP2C19
SCHEMBL7537438 0.88 CYP17A1 (0.65) CYP17A1CYP3A4CYP2C9CYP2C19
SCHEMBL7537443 0.88 CYP17A1 (0.65) CYP17A1CYP3A4CYP2C9CYP2C19
SCHEMBL4025212 0.88 CYP17A1 (0.65) CYP17A1CYP3A4CYP2C9CYP2C19
SCHEMBL4029239 0.87 CYP17A1 (0.66) CYP17A1CYP3A4HPGDSCYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1222174-B1 IMIDAZOL-4-YLMETHANOLS USED AS INHIBITORS OF STEROID C17-20 LYASE TAKEDA PHARMACEUTICAL (JP) 2009-05-27 EP disclosed
US-6713632-B1 Process for the preparation of imidazole derivatives TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2004-03-30 US disclosed
US-6649643-B1 Antitumor, anticarcinogenic, and antimetastasis agents; benign prostatic hyperplasia, alopecia, endometriosis, uterine myoma, hirsutism, virilism, precocious puberty, mastopathy, and polycystic overay syndrome treatment TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-11-18 US disclosed
EP-1222174-A1 IMIDAZOL-4-YLMETHANOLS USED AS INHIBITORS OF STEROID C17-20 LYASE Takeda Chemical Industries, Ltd. (JP) 2002-07-17 EP disclosed
EP-1193258-A1 PROCESS FOR THE PREPARATION OF IMIDAZOLE DERIVATIVES Takeda Chemical Industries, Ltd. (JP) 2002-04-03 EP disclosed
WO-2001030762-A1 IMIDAZOL-4-YLMETHANOLS USE AS INHIBITORS OF STEROID C17-20 LYASE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-03 WO disclosed