SCHEMBL4028778

SCHEMBL4028778

CC(C)C(O)(c1ccc2cc(C(=O)NCC(=O)O)ccc2c1)c1c[nH]cn1

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 15/20 0.54
CYP3A4 P08684 12/20 0.54
ATM Q13315 1/20 0.37
KDM4E B2RXH2 1/20 0.36
MAPT P10636 1/20 0.36
HIF1A Q16665 1/20 0.36
SLC22A6 Q4U2R8 1/20 0.36
SLC22A8 Q8TCC7 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
PTPRC P08575 2/20 0.36
CTSL P07711 1/20 0.36
PTPN13 Q12923 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4024213 0.90 CYP17A1 (0.67) CYP17A1CYP3A4
SCHEMBL4023743 0.90 CYP17A1 (0.67) CYP17A1CYP3A4
SCHEMBL7533841 0.89 CYP17A1 (0.53) CYP17A1CYP3A4KDM4E
SCHEMBL4027776 0.88 CYP17A1 (0.57) CYP17A1CYP3A4
SCHEMBL4025212 0.86 CYP17A1 (0.65) CYP17A1CYP3A4
SCHEMBL7537438 0.86 CYP17A1 (0.65) CYP17A1CYP3A4
SCHEMBL7537443 0.86 CYP17A1 (0.65) CYP17A1CYP3A4
SCHEMBL4025340 0.86 CYP17A1 (0.65) CYP17A1CYP3A4
SCHEMBL4026880 0.86 CYP17A1 (0.60) CYP17A1CYP3A4KDM4EMAPT
SCHEMBL4025132 0.85 CYP17A1 (0.66) CYP17A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1222174-B1 IMIDAZOL-4-YLMETHANOLS USED AS INHIBITORS OF STEROID C17-20 LYASE TAKEDA PHARMACEUTICAL (JP) 2009-05-27 EP disclosed
US-6649643-B1 Antitumor, anticarcinogenic, and antimetastasis agents; benign prostatic hyperplasia, alopecia, endometriosis, uterine myoma, hirsutism, virilism, precocious puberty, mastopathy, and polycystic overay syndrome treatment TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-11-18 US disclosed