SCHEMBL4025302

SCHEMBL4025302

CN1CCC(c2ncc(C(N)=O)s2)CC1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.41
GSK3B P49841 1/20 0.41
MLYCD O95822 1/20 0.40
HRH3 Q9Y5N1 1/20 0.39
SCD O00767 3/20 0.38
HTR1A P08908 2/20 0.37
HTR1D P28221 2/20 0.37
HTR1F P30939 2/20 0.37
JAK2 O60674 1/20 0.37
JAK1 P23458 1/20 0.37
JAK3 P52333 1/20 0.37
HTR1B P28222 1/20 0.37
MKNK1 Q9BUB5 1/20 0.36
WNT1 P04628 1/20 0.36
DYRK1A Q13627 1/20 0.36
PARP2 Q9UGN5 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21066432 0.86 GSK3B (0.41) GSK3BMLYCDHRH3SCDDYRK1A
SCHEMBL14164233 0.84 HDAC6 (0.46) HTR1AHTR1DHTR1FHTR1BMKNK1
SCHEMBL14164234 0.83 HRH3 (0.42) HRH3HTR1AHTR1DHTR1FHTR1B
SCHEMBL28312769 0.83 GSK3B (0.39) GSK3BMLYCDHRH3SCD
SCHEMBL628287 0.79 GSK3B (0.37) GSK3BMLYCDHRH3SCD
SCHEMBL14314254 0.74 ALOX15 (0.39) MLYCD
SCHEMBL628266 0.74 GSK3B (0.34) PARP1GSK3BMLYCDHRH3SCD
SCHEMBL23679874 0.74 SNCA (0.47)
SCHEMBL4781839 0.73 GSK3B (0.36) GSK3BMLYCDHRH3SCD
SCHEMBL12539166 0.73 TDP1 (0.35) MLYCDMKNK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2046793-A2 FUSED PYRIMIDO COMPOUNDS AstraZeneca AB (SE) 2009-04-15 EP disclosed
WO-2008003958-A2 FUSED PYRIMIDO COMPOUNDS ASTRAZENECA AB (SE) 2008-01-10 WO disclosed