SCHEMBL4025422

SCHEMBL4025422

Cc1ccc([N+](=O)[O-])c(C(=O)O)c1CCBr

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.53
TDP1 Q9NUW8 1/20 0.53
TSHR P16473 4/20 0.45
CES2 O00748 1/20 0.38
CES1 P23141 1/20 0.38
CASP6 P55212 1/20 0.38
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
HCAR3 P49019 1/20 0.37
MAPT P10636 3/20 0.36
MEN1 O00255 1/20 0.36
LMNA P02545 1/20 0.36
MAPK1 P28482 1/20 0.36
KMT2A Q03164 1/20 0.36
FBP1 P09467 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
POLB P06746 1/20 0.35
PKM P14618 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1613286 0.88 TDP1 (0.55) L3MBTL1TDP1TSHRCES2CES1
SCHEMBL27484681 0.81 TDP1 (0.36) L3MBTL1TDP1SMN1; SMN2MAPK1CA1
SCHEMBL27475187 0.80 TSHR (0.46) L3MBTL1TDP1TSHRSMN1; SMN2MAPT
SCHEMBL4025417 0.79 TDP1 (0.49) L3MBTL1TDP1TSHRCASP6NPC1
SCHEMBL20298737 0.76 TDP1 (0.60) L3MBTL1TDP1TSHRCES2CES1
SCHEMBL2257980 0.76 TDP1 (0.64) L3MBTL1TDP1TSHRCES2CES1
SCHEMBL3824611 0.76 TDP1 (0.64) L3MBTL1TDP1TSHRCES2CES1
SCHEMBL30527914 0.74 TDP1 (0.62) L3MBTL1TDP1TSHRCES2CES1
SCHEMBL21177973 0.74 TDP1 (0.62) L3MBTL1TDP1TSHRCES2CES1
SCHEMBL395027 0.74 TDP1 (0.62) L3MBTL1TDP1TSHRCES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102639498-A Process for preparing 2- (1-phenylethyl) isoindolin-1-one compounds CELGENE CORP 2012-08-15 CN disclosed
EP-2029535-A1 ISOINDOLE DERIVATIVES USEFUL FOR TREATING PAIN, GASTROINTESTINAL DISEASES AND CANCER AstraZeneca AB (SE) 2009-03-04 EP disclosed
WO-2007139464-A1 ISOINDOLE DERIVATIVES USEFUL FOR TREATING PAIN, GASTROINTESTINAL DISEASES AND CANCER ASTRAZENECA AB (SE) 2007-12-06 WO disclosed