SCHEMBL402764

SCHEMBL402764

COCOc1c(C)cc(C(=O)OC)cc1OC

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.50
PTPN1 P18031 1/20 0.44
KDM4E B2RXH2 3/20 0.44
CNR2 P34972 1/20 0.43
KMT2A Q03164 5/20 0.43
MEN1 O00255 3/20 0.43
ALDH1A1 P00352 2/20 0.42
MAPT P10636 3/20 0.42
PPARA Q07869 1/20 0.42
CYP3A4 P08684 1/20 0.42
HTT P42858 1/20 0.41
TPMT P51580 1/20 0.41
EGFR P00533 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
LMNA P02545 1/20 0.40
GAA P10253 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24425750 0.84 KMT2A (0.54) TSHRKDM4ECNR2KMT2AMEN1
SCHEMBL10205503 0.84 SMN1; SMN2 (0.53) TSHRPTPN1KDM4EKMT2AMEN1
SCHEMBL398872 0.84 BPTF (0.56) TSHRKDM4ECNR2KMT2AMEN1
SCHEMBL23202788 0.82 EGFR (0.48) TSHRPTPN1KDM4ECNR2KMT2A
SCHEMBL402919 0.82 KDM4E (0.42) TSHRPTPN1KDM4EALDH1A1MAPT
SCHEMBL400758 0.80 NOTUM (0.43) TSHRKDM4ECNR2KMT2AMEN1
SCHEMBL15341699 0.80 ALDH1A1 (0.55) TSHRKDM4EKMT2AMEN1ALDH1A1
SCHEMBL18018670 0.79 EGFR (0.48) TSHRKDM4ECNR2KMT2AMEN1
SCHEMBL10256166 0.79 EGFR (0.43) TSHRKDM4ECNR2ALDH1A1MAPT
SCHEMBL1739400 0.76 CA1 (0.54) TSHRKDM4ECNR2KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8101774-B2 Ester derivatives and medicinal use thereof JAPAN TOBACCO INC. (JP) 2012-01-24 US disclosed
US-8101774-B2 Ester derivatives and medicinal use thereof JAPAN TOBACCO INC. (JP) 2012-01-24 US disclosed
US-8101774-B2 Ester derivatives and medicinal use thereof JAPAN TOBACCO INC. (JP) 2012-01-24 US disclosed
EP-1803452-A1 ESTER DERIVATIVE AND PHARMACEUTICAL USE THEREOF Japan Tobacco, Inc. (JP) 2007-07-04 EP disclosed
US-20060089392-A1 Ester derivatives and medicinal use thereof JAPAN TOBACCO INC. (JP) 2006-04-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060089392-A1 Ester derivatives and medicinal use thereof MTTP, CETP, LIPA TSHR 1411/4885PTPN1 719/4885KDM4E 2908/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.