SCHEMBL4028632

SCHEMBL4028632

O=C(O)NCCc1ccc(-c2nn(C3CCCC3)c3c(F)cccc23)cc1

nearest known ligand 0.65

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.65
BTK Q06187 7/20 0.45
EGFR P00533 6/20 0.45
ALDH1A1 P00352 1/20 0.40
TSHR P16473 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
TAAR1 Q96RJ0 1/20 0.39
KCNJ6 P48051 1/20 0.39
KCNJ5 P48544 1/20 0.39
KCNJ3 P48549 1/20 0.39
TP53 P04637 1/20 0.39
CHRNA7 P36544 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4030596 0.87 ESR1 (0.69) ESR1BTKEGFR
SCHEMBL4028868 0.84 ESR1 (0.71) ESR1BTKEGFRKCNJ6KCNJ5
SCHEMBL27548056 0.80 ESR1 (0.62) ESR1BTKEGFR
SCHEMBL4027904 0.79 ESR1 (1.00) ESR1BTKEGFR
SCHEMBL27573495 0.78 ESR1 (0.61) ESR1BTKEGFRALDH1A1SMN1; SMN2
SCHEMBL4028037 0.78 ESR1 (0.61) ESR1BTKEGFR
SCHEMBL4028629 0.76 ESR1 (0.65) ESR1BTKEGFR
SCHEMBL4028322 0.76 ESR1 (0.71) ESR1EGFR
SCHEMBL4205205 0.75 ESR1 (0.73) ESR1BTKEGFR
SCHEMBL27548054 0.74 ESR1 (0.69) ESR1BTKEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1542976-B1 SUBSTITUTED 4-(INDAZOL-3-YL)PHENOLS AS ESTROGEN RECEPTOR (ER) LIGANDS AND THEIR USE IN THE TREATMENT OF INFLAMMATORY DISEASES WYETH CORP (US) 2009-02-04 EP claimed