SCHEMBL4028868

SCHEMBL4028868

O=C(O)Cc1ccc(-c2nn(C3CCCC3)c3c(F)cccc23)cc1

nearest known ligand 0.71

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.71
BTK Q06187 6/20 0.44
EGFR P00533 3/20 0.44
CMKLR1 Q99788 9/20 0.42
KCNJ6 P48051 1/20 0.41
KCNJ5 P48544 1/20 0.41
KCNJ3 P48549 1/20 0.41
ENPP2 Q13822 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4030596 0.89 ESR1 (0.69) ESR1BTKEGFRCMKLR1
SCHEMBL4028632 0.84 ESR1 (0.65) ESR1BTKEGFRKCNJ6KCNJ5
SCHEMBL4027904 0.83 ESR1 (1.00) ESR1BTKEGFRCMKLR1
SCHEMBL27548056 0.81 ESR1 (0.62) ESR1BTKEGFRCMKLR1
SCHEMBL4029342 0.81 ESR1 (0.69) ESR1BTKEGFRCMKLR1
SCHEMBL4028629 0.80 ESR1 (0.65) ESR1BTKEGFRCMKLR1
SCHEMBL4205205 0.79 ESR1 (0.73) ESR1BTKEGFR
SCHEMBL27548054 0.78 ESR1 (0.69) ESR1BTKEGFRCMKLR1
SCHEMBL4031188 0.78 ESR1 (0.72) ESR1BTKEGFRCMKLR1
SCHEMBL4027946 0.78 ESR1 (0.65) ESR1BTKEGFRCMKLR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1542976-B1 SUBSTITUTED 4-(INDAZOL-3-YL)PHENOLS AS ESTROGEN RECEPTOR (ER) LIGANDS AND THEIR USE IN THE TREATMENT OF INFLAMMATORY DISEASES WYETH CORP (US) 2009-02-04 EP claimed