SCHEMBL4028767

SCHEMBL4028767

Cc1noc(-c2ccc(COCC(=O)O)cc2)c1NC(=O)OC(c1ccccc1)C(F)(F)F

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LPAR1 Q92633 8/20 0.60
LPAR3 Q9UBY5 5/20 0.56
LPAR2 Q9HBW0 2/20 0.51
CYP2C9 P11712 2/20 0.49
ABCC3 O15438 1/20 0.49
ABCC4 O15439 1/20 0.49
ABCB11 O95342 1/20 0.49
CYP2C8 P10632 1/20 0.49
ABCB4 P21439 1/20 0.49
ABCC2 Q92887 1/20 0.49
SLCO1B3 Q9NPD5 1/20 0.49
SLCO1B1 Q9Y6L6 1/20 0.49
MAPT P10636 2/20 0.41
KDM4E B2RXH2 1/20 0.41
CYP3A4 P08684 1/20 0.34
GNRHR P30968 1/20 0.34
KLK7 P49862 1/20 0.33
ALDH1A1 P00352 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
RORC P51449 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4031915 0.92 LPAR1 (0.54) LPAR1LPAR3LPAR2CYP2C9ABCC3
SCHEMBL4028428 0.87 LPAR1 (0.61) LPAR1LPAR3LPAR2CYP2C9ABCC3
SCHEMBL4031913 0.85 LPAR1 (0.55) LPAR1LPAR3LPAR2CYP2C9ABCC3
SCHEMBL4033554 0.84 LPAR1 (0.68) LPAR1LPAR3LPAR2CYP2C9ABCC3
SCHEMBL4031685 0.82 LPAR1 (0.59) LPAR1LPAR3LPAR2CYP2C9ABCC3
SCHEMBL6374868 0.81 LPAR1 (0.60) LPAR1LPAR3LPAR2CYP2C9ABCC3
SCHEMBL4031090 0.80 LPAR1 (0.79) LPAR1LPAR3LPAR2CYP2C9ABCC3
SCHEMBL4029487 0.77 LPAR1 (0.48) LPAR1LPAR3LPAR2CYP2C9ABCC3
SCHEMBL16060770 0.75 LPAR1 (0.76) LPAR1LPAR3LPAR2CYP2C9ABCC3
SCHEMBL16060772 0.75 LPAR1 (0.76) LPAR1LPAR3LPAR2CYP2C9ABCC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1258484-B1 NOVEL ISOXAZOLE AND THIAZOLE COMPOUNDS AND USE THEREOF AS DRUGS KYOWA HAKKO KIRIN CO LTD (JP) 2009-01-14 EP claimed