SCHEMBL4029977

SCHEMBL4029977

CNC(=O)c1cc2ccc(C(O)(c3cn(C(c4ccccc4)(c4ccccc4)c4ccccc4)cn3)C(C)C)cc2cc1C

nearest known ligand 0.55

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 12/20 0.55
CYP3A4 P08684 11/20 0.55
SIRT2 Q8IXJ6 3/20 0.36
ACSS2 Q9NR19 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4033949 0.91 CYP3A4 (0.43) CYP17A1CYP3A4SIRT2
SCHEMBL1414920 0.89 CYP3A4 (0.42) CYP17A1CYP3A4SIRT2
SCHEMBL4025489 0.89 CYP3A4 (0.42) CYP17A1CYP3A4SIRT2
SCHEMBL4031099 0.89 CYP17A1 (0.52) CYP17A1CYP3A4SIRT2ACSS2
SCHEMBL4029531 0.87 CYP17A1 (0.56) CYP17A1CYP3A4SIRT2ACSS2
SCHEMBL4023981 0.85 CYP17A1 (0.42) CYP17A1CYP3A4SIRT2ACSS2
SCHEMBL7266948 0.84 CYP17A1 (0.56) CYP17A1CYP3A4SIRT2ACSS2
SCHEMBL1414954 0.84 CYP3A4 (0.39) CYP17A1CYP3A4SIRT2
SCHEMBL4026360 0.83 CYP3A4 (0.42) CYP17A1CYP3A4SIRT2ACSS2
SCHEMBL5750054 0.83 CYP3A4 (0.49) CYP17A1CYP3A4SIRT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1222174-B1 IMIDAZOL-4-YLMETHANOLS USED AS INHIBITORS OF STEROID C17-20 LYASE TAKEDA PHARMACEUTICAL (JP) 2009-05-27 EP disclosed
US-6649643-B1 Antitumor, anticarcinogenic, and antimetastasis agents; benign prostatic hyperplasia, alopecia, endometriosis, uterine myoma, hirsutism, virilism, precocious puberty, mastopathy, and polycystic overay syndrome treatment TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-11-18 US disclosed