SCHEMBL4030824

SCHEMBL4030824

CNC(=O)c1ccc2cc(C(O)(c3c[nH]cn3)C(C)C)ccc2c1C

nearest known ligand 0.68

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 19/20 0.68
CYP3A4 P08684 13/20 0.48
CYP2C8 P10632 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4030366 0.89 CYP17A1 (0.68) CYP17A1CYP3A4CYP2C8
SCHEMBL4023987 0.88 CYP17A1 (0.52) CYP17A1CYP3A4CYP2C8
SCHEMBL4024772 0.87 CYP17A1 (0.51) CYP17A1CYP3A4
SCHEMBL4030338 0.85 CYP17A1 (0.67) CYP17A1CYP3A4
SCHEMBL4030837 0.84 CYP17A1 (0.48) CYP17A1CYP3A4CYP2C8
SCHEMBL4025340 0.82 CYP17A1 (0.65) CYP17A1CYP3A4
SCHEMBL7537443 0.82 CYP17A1 (0.65) CYP17A1CYP3A4
SCHEMBL7537438 0.82 CYP17A1 (0.65) CYP17A1CYP3A4
SCHEMBL4025212 0.82 CYP17A1 (0.65) CYP17A1CYP3A4
SCHEMBL4027111 0.82 CYP17A1 (0.46) CYP17A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1222174-B1 IMIDAZOL-4-YLMETHANOLS USED AS INHIBITORS OF STEROID C17-20 LYASE TAKEDA PHARMACEUTICAL (JP) 2009-05-27 EP disclosed
US-6649643-B1 Antitumor, anticarcinogenic, and antimetastasis agents; benign prostatic hyperplasia, alopecia, endometriosis, uterine myoma, hirsutism, virilism, precocious puberty, mastopathy, and polycystic overay syndrome treatment TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-11-18 US disclosed