SCHEMBL4030998

SCHEMBL4030998

CC(C)C(O)(c1ccc2c(Cl)c(O[Si](C)(C)C(C)(C)C)ccc2c1)c1cn(C(c2ccccc2)(c2ccccc2)c2ccccc2)cn1

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
RORC P51449 3/20 0.36
CYP3A4 P08684 9/20 0.34
CYP17A1 P05093 6/20 0.33
CYP2C9 P11712 2/20 0.32
CYP2C19 P33261 2/20 0.32
SIRT2 Q8IXJ6 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1415016 0.91 CYP3A4 (0.34) RORCCYP3A4CYP17A1CYP2C9CYP2C19
SCHEMBL4028814 0.86 CYP17A1 (0.36) CYP3A4CYP17A1SIRT2
SCHEMBL1414804 0.86 CYP17A1 (0.38) CYP3A4CYP17A1CYP2C9CYP2C19SIRT2
SCHEMBL1414831 0.85 CYP3A4 (0.40) CYP3A4CYP17A1CYP2C9CYP2C19SIRT2
SCHEMBL4032165 0.85 RORC (0.40) RORCCYP3A4CYP17A1CYP2C9CYP2C19
SCHEMBL4030196 0.84 RORC (0.35) RORCCYP3A4CYP17A1CYP2C9CYP2C19
SCHEMBL4026083 0.82 CYP17A1 (0.44) RORCCYP3A4CYP17A1SIRT2
SCHEMBL4030722 0.81 RORC (0.41) RORCCYP3A4CYP17A1SIRT2
SCHEMBL4023660 0.81 RORC (0.38) RORCCYP3A4CYP17A1SIRT2
SCHEMBL4027150 0.81 CYP17A1 (0.44) RORCCYP3A4CYP17A1SIRT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1222174-B1 IMIDAZOL-4-YLMETHANOLS USED AS INHIBITORS OF STEROID C17-20 LYASE TAKEDA PHARMACEUTICAL (JP) 2009-05-27 EP disclosed
US-6649643-B1 Antitumor, anticarcinogenic, and antimetastasis agents; benign prostatic hyperplasia, alopecia, endometriosis, uterine myoma, hirsutism, virilism, precocious puberty, mastopathy, and polycystic overay syndrome treatment TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-11-18 US disclosed
EP-1222174-A1 IMIDAZOL-4-YLMETHANOLS USED AS INHIBITORS OF STEROID C17-20 LYASE Takeda Chemical Industries, Ltd. (JP) 2002-07-17 EP disclosed
WO-2001030762-A1 IMIDAZOL-4-YLMETHANOLS USE AS INHIBITORS OF STEROID C17-20 LYASE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-03 WO disclosed