SCHEMBL4033491

SCHEMBL4033491

CN1CCC(Oc2cc(O)cc3ncnc(Nc4ccc(F)c(Cl)c4)c23)CC1

nearest known ligand 0.79

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EGFR P00533 19/20 0.79
ERBB2 P04626 4/20 0.62
KCNH2 Q12809 1/20 0.57
SRC P12931 1/20 0.55
HPGD P15428 1/20 0.53
HTT P42858 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL4033517 0.94 EGFR (0.70) EGFRERBB2KCNH2SRC
SCHEMBL4034609 0.89 EGFR (1.00) EGFRERBB2SRC
SCHEMBL4213030 0.87 EGFR (0.77) EGFRERBB2
SCHEMBL4040179 0.87 EGFR (1.00) EGFRERBB2KCNH2SRC
SCHEMBL4034340 0.86 EGFR (0.83) EGFRERBB2KCNH2SRC
SCHEMBL4036009 0.85 EGFR (0.81) EGFRERBB2KCNH2SRC
SCHEMBL4031827 0.85 EGFR (0.81) EGFRERBB2KCNH2SRC
SCHEMBL4037607 0.85 EGFR (0.84) EGFRERBB2KCNH2
SCHEMBL4032825 0.85 EGFR (0.78) EGFRERBB2KCNH2SRC
SCHEMBL4036214 0.85 EGFR (0.83) EGFRERBB2KCNH2SRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1444211-B1 QUINAZOLINE DERIVATIVES AS ANTITUMOR AGENTS ASTRAZENECA AB (SE) 2009-01-21 EP disclosed