SCHEMBL4033873

SCHEMBL4033873

CN1CCC(Oc2cc(OCCCN3CCOCC3)cc3ncnc(Nc4ccc(F)c(Cl)c4)c23)CC1

nearest known ligand 0.89

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 12/20 0.89
SRC P12931 9/20 0.65
KDR P35968 9/20 0.65
CIT O14578 1/20 0.60
GAK O14976 1/20 0.60
EPHB6 O15197 1/20 0.60
ABCC4 O15439 1/20 0.60
DAPK3 O43293 1/20 0.60
RIPK2 O43353 1/20 0.60
NR1I2 O75469 1/20 0.60
RPS6KA4 O75676 1/20 0.60
STK17B O94768 1/20 0.60
STK10 O94804 1/20 0.60
PRKD3 O94806 1/20 0.60
ABCB11 O95342 1/20 0.60
MAP4K4 O95819 1/20 0.60
CHEK2 O96017 1/20 0.60
ABL1 P00519 1/20 0.60
ERBB2 P04626 1/20 0.60
LCK P06239 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4035070 0.96 EGFR (0.82) EGFRSRCKDRGAKEPHB6
SCHEMBL4037393 0.96 EGFR (0.84) EGFRSRCKDRGAKEPHB6
SCHEMBL4036758 0.95 EGFR (0.90) EGFRSRCKDRCITGAK
SCHEMBL4035967 0.94 EGFR (1.00) EGFRSRCKDRGAKEPHB6
SCHEMBL4036399 0.94 EGFR (0.91) EGFRSRCKDRCITGAK
SCHEMBL4041510 0.94 EGFR (0.84) EGFRSRCKDRCITGAK
SCHEMBL4037323 0.94 EGFR (0.89) EGFRSRCKDRERBB2
SCHEMBL4037159 0.93 EGFR (0.85) EGFRSRCKDRCITGAK
SCHEMBL4037082 0.93 EGFR (0.82) EGFRSRCKDRLCK
SCHEMBL4031704 0.93 EGFR (0.81) EGFRSRCKDRLCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1444211-B1 QUINAZOLINE DERIVATIVES AS ANTITUMOR AGENTS ASTRAZENECA AB (SE) 2009-01-21 EP disclosed