SCHEMBL4035824

SCHEMBL4035824

Cc1cnc(CN(Cc2ncccc2C(C)(C)c2ccc(F)cc2)C2CCN(C(=O)c3ncc[nH]3)CC2)c(C)c1

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.35
HTR2B P41595 2/20 0.35
CCR3 P51677 4/20 0.34
CXCR4 P61073 2/20 0.34
RBP4 P02753 1/20 0.33
SMO Q99835 1/20 0.33
RORC P51449 1/20 0.33
TYRO3 Q06418 1/20 0.32
TRPV1 Q8NER1 1/20 0.32
POLB P06746 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2084734 0.88 TRPV1 (0.38) CYP3A4CXCR4TRPV1
SCHEMBL5051530 0.88 SMO (0.36) CYP3A4CCR3CXCR4SMOTRPV1
SCHEMBL23428751 0.87 CXCR4 (0.36) CYP3A4CCR3CXCR4SMOTRPV1
SCHEMBL2084270 0.86 CXCR4 (0.40) HTR2BCXCR4SMOTYRO3
SCHEMBL2084834 0.86 TRPV1 (0.38) CYP3A4CCR3CXCR4SMOTRPV1
SCHEMBL2083669 0.85 MEN1 (0.44)
SCHEMBL2082435 0.83 FAAH (0.38) CYP3A4CCR3CXCR4SMOTRPV1
SCHEMBL2084322 0.82 TRPV1 (0.36) RBP4TRPV1
SCHEMBL5053640 0.82 CXCR4 (0.37) CYP3A4CXCR4RBP4SMOTRPV1
SCHEMBL2082075 0.81 CXCR4 (0.38) CXCR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1613613-A4 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC (CA) 2009-03-25 EP disclosed
EP-1613613-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2006-01-11 EP disclosed
WO-2004091518-A2 CXCR4 CHEMOKINE RECEPTOR BINDING COMPOUNDS ANORMED INC. (CA) 2004-10-28 WO disclosed