SCHEMBL4036035

SCHEMBL4036035

CC(C)(C)N(C(=O)O)S(=O)(=O)c1nnc(-c2ccc(OCCCCl)cc2)s1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 3/20 0.43
HDAC2 Q92769 3/20 0.43
HDAC6 Q9UBN7 1/20 0.42
MAPT P10636 4/20 0.41
RAB9A P51151 3/20 0.41
LMNA P02545 1/20 0.41
XIAP P98170 1/20 0.41
NR1H4 Q96RI1 1/20 0.40
KDM4E B2RXH2 4/20 0.39
NPC1 O15118 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
TP53 P04637 4/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
HSD17B10 Q99714 3/20 0.35
CSNK2A2 P19784 1/20 0.35
CSNK2A1 P68400 1/20 0.35
ALDH1A1 P00352 1/20 0.35
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3484094 0.78 XIAP (0.36) HDAC1HDAC2HDAC6MAPTRAB9A
SCHEMBL3483775 0.78 HDAC1 (0.48) HDAC1HDAC2HDAC6MAPTRAB9A
SCHEMBL3483840 0.77 RAB9A (0.50) HDAC1HDAC2HDAC6MAPTRAB9A
SCHEMBL3483727 0.75 RAB9A (0.43) HDAC1HDAC2HDAC6MAPTRAB9A
SCHEMBL3483730 0.75 RAB9A (0.43) HDAC1HDAC2HDAC6MAPTRAB9A
SCHEMBL3483445 0.73 HDAC1 (0.46) HDAC1HDAC2HDAC6MAPTRAB9A
SCHEMBL3483079 0.72 RAB9A (0.47) HDAC1HDAC2HDAC6MAPTRAB9A
SCHEMBL3484166 0.71 RAB9A (0.41) HDAC1HDAC2HDAC6MAPTRAB9A
SCHEMBL3483720 0.71 HDAC1 (0.41) HDAC1HDAC2HDAC6MAPTRAB9A
SCHEMBL3483333 0.70 KDM4E (0.41) HDAC1HDAC2HDAC6MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049200-A2 NOVEL INHIBITORS OF BETA-LACTAMASE MethylGene Inc. (CA) 2009-04-22 EP disclosed
WO-2008073142-A2 NOVEL INHIBITORS OF BETA-LACTAMASE MERCK & CO., INC. (US) 2008-06-19 WO disclosed