SCHEMBL4036831

SCHEMBL4036831

COc1cc2ncn(C3=CC(OCc4cccs4)C(=S)C(C#N)=C3)c2cc1OC

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 7/20 0.46
IKBKE Q14164 11/20 0.41
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 2/20 0.40
LMNA P02545 2/20 0.40
MAPT P10636 2/20 0.40
HPGD P15428 2/20 0.40
TDP1 Q9NUW8 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
GPR55 Q9Y2T6 1/20 0.40
FGFR1 P11362 1/20 0.38
SRC P12931 1/20 0.38
TBK1 Q9UHD2 1/20 0.38
NPC1 O15118 1/20 0.37
ALOX15 P16050 1/20 0.37
TSHR P16473 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
GAA P10253 1/20 0.35
KIT P10721 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4035304 0.85 PLK1 (0.46) PLK1IKBKEFGFR1SRCTBK1
SCHEMBL4040575 0.84 IKBKE (0.40) PLK1IKBKEFGFR1SRCTBK1
SCHEMBL4040312 0.83 IKBKE (0.42) PLK1IKBKEFGFR1SRCTBK1
SCHEMBL4032649 0.82 IKBKE (0.39) PLK1IKBKEFGFR1SRCTBK1
SCHEMBL4034367 0.81 PLK1 (0.44) PLK1IKBKEFGFR1SRCTBK1
SCHEMBL4032684 0.81 FGFR1 (0.43) PLK1IKBKEFGFR1SRCTBK1
SCHEMBL4034652 0.81 PLK1 (0.57) PLK1IKBKEFGFR1SRCTBK1
SCHEMBL4033043 0.81 PLK1 (0.48) PLK1IKBKEFGFR1SRCTBK1
SCHEMBL4035204 0.80 IKBKE (0.38) PLK1IKBKEFGFR1SRCTBK1
SCHEMBL4037133 0.79 IKBKE (0.37) PLK1IKBKEFGFR1SRCTBK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720864-B1 BENZIMIDAZOL SUBSTITUTED THIOPHENE DERIVATIVES WITH ACTIVITY ON IKK3 GLAXO GROUP LTD (GB) 2009-05-06 EP claimed