SCHEMBL4037270

SCHEMBL4037270

C=CCNC(=O)[C@H]1CN(C(=O)OC(C)(C)C)CCN1S(=O)(=O)c1cccc2cccnc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.51
HPGD P15428 1/20 0.51
GAA P10253 3/20 0.48
POLB P06746 2/20 0.48
MAPT P10636 3/20 0.47
LMNA P02545 2/20 0.47
USP2 O75604 1/20 0.47
HTT P42858 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
TSHR P16473 2/20 0.47
GFER P55789 1/20 0.47
HCRTR1 O43613 1/20 0.47
KMT2A Q03164 1/20 0.47
ATM Q13315 1/20 0.46
MMP1 P03956 1/20 0.45
MMP3 P08254 1/20 0.45
MMP7 P09237 1/20 0.45
MMP9 P14780 1/20 0.45
TP53 P04637 2/20 0.45
HSP90AA1 P07900 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14499802 1.00 ALDH1A1 (0.51) ALDH1A1HPGDGAAPOLBMAPT
SCHEMBL4037427 0.88 TSHR (0.52) ALDH1A1HPGDGAAPOLBMAPT
SCHEMBL1380179 0.84 GAA (0.51) ALDH1A1HPGDGAAPOLBMAPT
SCHEMBL13886846 0.84 GAA (0.51) ALDH1A1HPGDGAAPOLBMAPT
Hydrochloric Acid SCHEMBL4035609 0.83 GAA (0.50) ALDH1A1HPGDGAAPOLBMAPT
Hydrochloric Acid SCHEMBL4034494 0.83 GAA (0.50) ALDH1A1HPGDGAAPOLBMAPT
SCHEMBL4035463 0.83 GAA (0.53) ALDH1A1HPGDGAAPOLBMAPT
SCHEMBL4033037 0.82 SMN1; SMN2 (0.49) ALDH1A1HPGDGAAPOLBMAPT
Hydrochloric Acid SCHEMBL4365526 0.82 ALDH1A1 (0.49) ALDH1A1HPGDGAAPOLBMAPT
SCHEMBL4035900 0.82 SMN1; SMN2 (0.49) ALDH1A1HPGDGAAPOLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1592389-B1 PIPERAZINE-2-CARBOXAMIDE DERIVATIVES SERONO LAB (CH) 2009-04-22 EP claimed