SCHEMBL4037394

SCHEMBL4037394

Cc1cccc(Nc2ncnc3cc(O)cc(OC4CCN(C)CC4)c23)c1

nearest known ligand 0.57

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EGFR P00533 13/20 0.57
ERBB2 P04626 4/20 0.57
KCNH2 Q12809 1/20 0.53
SRC P12931 6/20 0.51
KDR P35968 3/20 0.51
MKNK1 Q9BUB5 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL4039319 0.93 EGFR (0.53) EGFRERBB2KCNH2SRCKDR
SCHEMBL4031239 0.88 EGFR (0.71) EGFRERBB2KCNH2SRCKDR
Hydrochloric Acid SCHEMBL4034029 0.87 EGFR (0.70) EGFRERBB2KCNH2SRCKDR
SCHEMBL4036988 0.85 EGFR (0.56) EGFRERBB2KCNH2SRCKDR
SCHEMBL4046007 0.84 EGFR (0.59) EGFRERBB2KCNH2SRCKDR
Trifluoroacetic Acid SCHEMBL4032839 0.83 EGFR (0.58) EGFRERBB2KCNH2SRCKDR
Trifluoroacetic Acid SCHEMBL4034846 0.83 EGFR (0.52) EGFRERBB2KCNH2SRCKDR
SCHEMBL4039322 0.83 EGFR (0.56) EGFRERBB2KCNH2SRCKDR
SCHEMBL4033491 0.83 EGFR (0.79) EGFRERBB2KCNH2SRC
SCHEMBL5406753 0.80 EGFR (0.73) EGFRERBB2KCNH2SRCKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1444211-B1 QUINAZOLINE DERIVATIVES AS ANTITUMOR AGENTS ASTRAZENECA AB (SE) 2009-01-21 EP disclosed