SCHEMBL4038722

SCHEMBL4038722

Nc1nc(Nc2ccccc2)nn1-c1cc(NC(CO)c2ccccc2)ncn1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
FLT3 P36888 12/20 0.44
KIT P10721 8/20 0.44
IRAK4 Q9NWZ3 3/20 0.44
AURKA O14965 2/20 0.44
JAK3 P52333 1/20 0.42
AXL P30530 2/20 0.38
JAK2 O60674 1/20 0.38
EGFR P00533 3/20 0.38
NPSR1 Q6W5P4 1/20 0.37
RPS6KB1 P23443 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12780393 1.00 FLT3 (0.44) FLT3KITIRAK4AURKAJAK3
SCHEMBL12780389 1.00 FLT3 (0.44) FLT3KITIRAK4AURKAJAK3
SCHEMBL12780487 0.92 FLT3 (0.43) FLT3KITIRAK4AURKAJAK3
SCHEMBL4042917 0.92 FLT3 (0.43) FLT3KITIRAK4AURKAJAK3
SCHEMBL12781173 0.90 CDK1 (0.46) FLT3KITAURKAJAK3AXL
SCHEMBL4042422 0.90 FLT3 (0.46) FLT3KITIRAK4AURKAJAK3
SCHEMBL12780482 0.90 FLT3 (0.46) FLT3KITIRAK4AURKAJAK3
SCHEMBL12780484 0.90 FLT3 (0.46) FLT3KITIRAK4AURKAJAK3
SCHEMBL4038537 0.89 FLT3 (0.46) FLT3KITIRAK4AURKAJAK3
SCHEMBL12780516 0.87 FLT3 (0.47) FLT3KITIRAK4AURKAAXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1562589-B1 DIAMINOTRIAZOLES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMA (US) 2009-01-07 EP disclosed