SCHEMBL4039332

SCHEMBL4039332

CC(C)CC(NC(=O)c1ccc(N)cc1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)c1ccc[n+]([O-])c1

nearest known ligand 0.53

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CTSK P43235 11/20 0.53
CTSS P25774 3/20 0.42
CA1 P00915 3/20 0.39
CA2 P00918 2/20 0.39
CA12 O43570 2/20 0.37
CA9 Q16790 2/20 0.37
CCR1 P32246 1/20 0.37
CTSV O60911 2/20 0.36
CTSL P07711 2/20 0.36
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4042980 0.94 CTSK (0.53) CTSKCTSSCA1CA2CA12
SCHEMBL4038667 0.93 CTSK (0.54) CTSKCTSSCA1CA2CCR1
SCHEMBL4042230 0.93 CTSK (0.52) CTSKCTSSCA1CA2CA12
SCHEMBL4040650 0.92 CTSK (0.65) CTSKCTSSCA1CA2CA12
SCHEMBL4039127 0.91 CTSK (0.61) CTSKCTSSCA1CA2CCR1
SCHEMBL4044649 0.91 CTSK (0.65) CTSKCTSSCA1CA2CA12
SCHEMBL4042967 0.91 CTSK (0.52) CTSKCTSSCA2CTSLPOLB
SCHEMBL4045969 0.91 CTSK (0.56) CTSKCTSSCA1CA2CCR1
SCHEMBL4040991 0.91 CTSK (0.52) CTSKCTSSCA1CA2CCR1
SCHEMBL4044521 0.90 CTSK (0.51) CTSKCTSSCA1CA2CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed
EP-1651592-B1 NOVEL DIBENZO[B,F]OXEPINE-10-CARBOXAMIDES AND PHARMACEUTICAL USES THEREOF NOVARTIS AG (CH) 2009-04-29 EP disclosed