SCHEMBL4042895

SCHEMBL4042895

CC(=O)NC(C(=O)N1CC(=O)C2C1CCN2C(=O)C(CC(C)C)NC(=O)Oc1ccc(-c2ccccc2)s1)C(C)(C)C

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CTSK P43235 14/20 0.51
CTSS P25774 6/20 0.38
CTSL P07711 7/20 0.37
CTSB P07858 2/20 0.37
MAPK1 P28482 1/20 0.35
ACE2 Q9BYF1 1/20 0.35
CASP1 P29466 1/20 0.33
CASP3 P42574 1/20 0.33
CASP2 P42575 1/20 0.33
CASP4 P49662 1/20 0.33
CASP5 P51878 1/20 0.33
CASP7 P55210 1/20 0.33
CASP9 P55211 1/20 0.33
CASP8 Q14790 1/20 0.33
CASP10 Q92851 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4049584 0.93 CTSK (0.51) CTSKCTSSCTSLCTSBMAPK1
SCHEMBL4047665 0.92 CTSK (0.51) CTSKCTSSCTSLCTSBMAPK1
SCHEMBL4047203 0.91 CTSK (0.48) CTSKCTSSCTSLCTSBACE2
SCHEMBL4043538 0.91 CTSK (0.49) CTSKCTSSCTSLCTSBMAPK1
SCHEMBL4047843 0.90 CTSK (0.49) CTSKCTSSCTSLCTSBMAPK1
SCHEMBL4039890 0.90 CTSK (0.48) CTSKCTSSCTSLCTSBMAPK1
SCHEMBL4048373 0.90 CTSK (0.52) CTSKCTSSCTSLCTSBMAPK1
SCHEMBL4051840 0.89 CTSK (0.48) CTSKCTSSCTSLCTSBACE2
SCHEMBL4045644 0.89 CTSK (0.51) CTSKCTSSCTSLCTSBMAPK1
SCHEMBL4044409 0.89 CTSK (0.50) CTSKCTSSCTSLCTSBMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed