SCHEMBL4042930

SCHEMBL4042930

Cc1ccccc1Nc1nc(N)n(-c2ncccc2I)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FLT3 P36888 7/20 0.48
IRAK4 Q9NWZ3 4/20 0.48
KIT P10721 4/20 0.48
AURKA O14965 2/20 0.48
HTT P42858 2/20 0.44
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
NTSR1 P30989 1/20 0.41
CYP2C19 P33261 1/20 0.41
KMT2A Q03164 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
CCNB2 O95067 1/20 0.40
CDK1 P06493 1/20 0.40
RET P07949 1/20 0.40
CCNB1 P14635 1/20 0.40
CCNB3 Q8WWL7 1/20 0.40
LMNA P02545 2/20 0.39
ALDH1A1 P00352 2/20 0.39
GAA P10253 2/20 0.39
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12779700 0.80 FLT3 (0.73) FLT3IRAK4KITAURKAHTT
SCHEMBL12845286 0.75 FLT3 (0.73) FLT3IRAK4KITAURKAAXL
SCHEMBL4046948 0.73 FLT3 (0.48) FLT3IRAK4KITAURKAKMT2A
SCHEMBL12845470 0.70 FLT3 (0.61) FLT3IRAK4KITAURKAAXL
SCHEMBL12845662 0.69 FLT3 (0.63) FLT3IRAK4KITAURKAKMT2A
SCHEMBL12780242 0.68 FLT3 (0.53) FLT3IRAK4KITAURKAHTT
SCHEMBL3950995 0.68 HTT (0.56) HTTCYP3A4CYP2C9NTSR1CYP2C19
SCHEMBL4040866 0.68 FLT3 (0.67) FLT3IRAK4KITAURKAALDH1A1
SCHEMBL4042831 0.67 FLT3 (0.60) FLT3IRAK4KITAURKAPTK2
SCHEMBL4039960 0.66 FLT3 (0.67) FLT3IRAK4KITAURKAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1562589-B1 DIAMINOTRIAZOLES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMA (US) 2009-01-07 EP disclosed