SCHEMBL4043104

SCHEMBL4043104

CC(=O)NC(C(=O)N1CC(=O)C2C1CCN2C(=O)C(CC(C)C)NC(=O)Oc1ccc(-c2ccccc2)s1)C1CCCC1

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CTSK P43235 15/20 0.47
CTSL P07711 8/20 0.37
CTSS P25774 8/20 0.37
CTSB P07858 2/20 0.37
CTSV O60911 1/20 0.36
ACE2 Q9BYF1 2/20 0.36
MMP1 P03956 1/20 0.35
MMP13 P45452 1/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4042551 0.99 CTSK (0.47) CTSKCTSLCTSSCTSBCTSV
SCHEMBL4049584 0.93 CTSK (0.51) CTSKCTSLCTSSCTSBACE2
SCHEMBL4043538 0.91 CTSK (0.49) CTSKCTSLCTSSCTSBACE2
SCHEMBL4044504 0.90 CTSK (0.48) CTSKCTSLCTSSCTSBMEN1
SCHEMBL4047843 0.90 CTSK (0.49) CTSKCTSLCTSSCTSBACE2
SCHEMBL4041776 0.90 CTSK (0.47) CTSKCTSLCTSSCTSBCTSV
SCHEMBL4047203 0.90 CTSK (0.48) CTSKCTSLCTSSCTSBACE2
SCHEMBL4039890 0.90 CTSK (0.48) CTSKCTSLCTSSCTSBACE2
SCHEMBL4047665 0.89 CTSK (0.51) CTSKCTSLCTSSCTSBACE2
SCHEMBL4051840 0.89 CTSK (0.48) CTSKCTSLCTSSCTSBACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed