SCHEMBL4043637

SCHEMBL4043637

COc1ccc(C2(C(C(=O)NC(C)(C)C)C3CCCCC3)Nc3ccccc3N2)c(OC)c1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.41
ALDH1A1 P00352 3/20 0.41
NPC1 O15118 2/20 0.41
MAPT P10636 1/20 0.41
MEN1 O00255 4/20 0.40
KMT2A Q03164 4/20 0.40
LPAR1 Q92633 2/20 0.38
METAP2 P50579 2/20 0.38
METAP1 P53582 1/20 0.38
TAS1R3 Q7RTX0 1/20 0.37
TAS1R1 Q7RTX1 1/20 0.37
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NFKB1 P19838 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1577410 0.89 MEN1 (0.48) RAB9AALDH1A1NPC1MAPTMEN1
SCHEMBL4034697 0.89 MEN1 (0.48) RAB9AALDH1A1NPC1MAPTMEN1
SCHEMBL4044757 0.89 MEN1 (0.48) RAB9AALDH1A1NPC1MAPTMEN1
SCHEMBL4035037 0.87 ALDH1A1 (0.50) RAB9AALDH1A1NPC1MAPTMEN1
SCHEMBL4040175 0.85 KMT2A (0.50) RAB9AALDH1A1NPC1MAPTMEN1
SCHEMBL4044363 0.84 ALDH1A1 (0.41) RAB9AALDH1A1NPC1MAPTMEN1
SCHEMBL4039125 0.84 MEN1 (0.42) RAB9AALDH1A1NPC1MAPTMEN1
SCHEMBL4040874 0.84 PTPN1 (0.44) RAB9AALDH1A1NPC1MAPTMEN1
SCHEMBL4043980 0.84 ALDH1A1 (0.41) RAB9AALDH1A1NPC1MAPTMEN1
SCHEMBL4035711 0.83 TSHR (0.42) RAB9AALDH1A1NPC1MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2038259-A1 BENZIMIDAZOLE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF, THEIR USE AS FXR AGONISTS AND PHARMACEUTICAL PREPARATIONS CONTAINING THE SAME F.HOFFMANN-LA ROCHE AG (CH) 2009-03-25 EP disclosed
WO-2008000643-A1 BENZIMIDAZOLE DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF, THEIR USE AS FXR AGONISTS AND PHARMACEUTICAL PREPARATIONS CONTAINING THE SAME F. HOFFMANN-LA ROCHE AG (CH) 2008-01-03 WO disclosed