SCHEMBL4044276

SCHEMBL4044276

O=C1NC(=S)NC(=O)C1=CC=Cc1ccccc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
METAP1 P53582 4/20 1.00
ALDH1A1 P00352 6/20 0.73
RAB9A P51151 2/20 0.73
MAPT P10636 9/20 0.62
APP P05067 2/20 0.62
SNCA P37840 2/20 0.62
F2 P00734 1/20 0.59
MEN1 O00255 5/20 0.57
KMT2A Q03164 5/20 0.57
MAPK1 P28482 4/20 0.57
POLB P06746 3/20 0.57
PKM P14618 2/20 0.57
LMNA P02545 2/20 0.57
NTSR1 P30989 2/20 0.57
NPSR1 Q6W5P4 2/20 0.57
KDM4E B2RXH2 1/20 0.57
L3MBTL1 Q9Y468 1/20 0.57
CMA1 P23946 1/20 0.56
MITF O75030 2/20 0.56
SMN1; SMN2 Q16637 2/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13848519 1.00 METAP1 (1.00) METAP1ALDH1A1RAB9AMAPTAPP
SCHEMBL11598594 0.86 METAP1 (1.00) METAP1ALDH1A1RAB9AMAPTAPP
SCHEMBL11598589 0.86 METAP1 (1.00) METAP1ALDH1A1RAB9AMAPTAPP
SCHEMBL14712875 0.83 METAP1 (0.71) METAP1ALDH1A1RAB9AMAPTAPP
SCHEMBL14712988 0.83 METAP1 (0.71) METAP1ALDH1A1RAB9AMAPTAPP
SCHEMBL14713019 0.82 METAP1 (0.68) METAP1ALDH1A1RAB9AMAPTAPP
SCHEMBL16543021 0.82 METAP1 (0.68) METAP1ALDH1A1RAB9AMAPTAPP
SCHEMBL14713027 0.80 MAPT (0.77) METAP1ALDH1A1RAB9AMAPTAPP
SCHEMBL8026269 0.80 METAP1 (1.00) METAP1ALDH1A1RAB9AMAPTAPP
SCHEMBL14712871 0.80 METAP1 (0.66) METAP1ALDH1A1RAB9AMAPTAPP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1305026-B1 BARBITURIC ACID ANALOGS AS THERAPEUTIC AGENTS NOVUSPHARMA SPA (IT) 2009-05-13 EP disclosed
US-20080113993-A1 BARBITURIC ACID ANALOGS AS THERAPEUTIC AGENTS VIA ARIOSTO, 23 (IT) 2008-05-15 US disclosed
US-20030229108-A1 Barbituric acid analogs as therapeutic agents NOVUSPHARMA S.P.A. (IT) 2003-12-11 US disclosed
EP-1305026-A2 BARBITURIC ACID ANALOGS AS THERAPEUTIC AGENTS Novuspharma S.p.A. (IT) 2003-05-02 EP disclosed
WO-2001093841-A2 BARBITURIC ACID ANALOGS AS THERAPEUTIC AGENTS NOVUSPHARMA S.P.A. (IT) 2001-12-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030229108-A1 Barbituric acid analogs as therapeutic agents HIF1AN, HIF1A, VHL METAP1 2079/4885ALDH1A1 123/4885RAB9A 4155/4885
US-20080113993-A1 BARBITURIC ACID ANALOGS AS THERAPEUTIC AGENTS HIF1A, HIF1AN, PDGFA METAP1 2162/4885ALDH1A1 93/4885RAB9A 3153/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.