SCHEMBL4045973

SCHEMBL4045973

COc1ccc(C(F)C=O)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.48
CYP2A6 P11509 1/20 0.48
CA1 P00915 2/20 0.46
CA2 P00918 2/20 0.46
CA12 O43570 1/20 0.46
CA7 P43166 1/20 0.46
CA9 Q16790 1/20 0.46
CA14 Q9ULX7 1/20 0.46
TSHR P16473 1/20 0.44
MAPK1 P28482 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
ACP3 P15309 1/20 0.42
SLC2A1 P11166 1/20 0.41
ACHE P22303 2/20 0.41
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C19 P33261 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
MEN1 O00255 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4775938 0.78 ALDH1A1 (0.52) ALDH1A1CYP2A6CA1CA2CA12
SCHEMBL182145 0.78 ALDH1A1 (0.52) ALDH1A1CYP2A6CA1CA2CA12
SCHEMBL22498336 0.77 CHRM2 (0.49) ALDH1A1CA1CA2CA7CA9
SCHEMBL615428 0.77 ALDH1A1 (0.50) ALDH1A1CYP2A6CA1CA2CA12
SCHEMBL11324732 0.76 CYP2A6 (0.42) ALDH1A1CYP2A6CA1CA2CA12
SCHEMBL23540648 0.75 ALDH1A1 (0.48) ALDH1A1CYP2A6CA1CA2CA12
SCHEMBL1155920 0.75 ALDH1A1 (0.48) ALDH1A1CYP2A6CA1CA2CA12
SCHEMBL29207873 0.75 ALDH1A1 (0.48) ALDH1A1CYP2A6CA1CA2CA12
SCHEMBL2591240 0.75 ALDH1A1 (0.48) ALDH1A1CYP2A6CA1CA2CA12
SCHEMBL6194589 0.75 ALDH1A1 (0.48) ALDH1A1CYP2A6CA1CA2CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2026799-A2 IMIDAZOLIDINE DERIVATIVES, USES THEREFOR, PREPARATION THEREOF AND COMPOSITIONS COMPRISING SUCH Galapagos SAS (FR) 2009-02-25 EP disclosed
WO-2008134036-A1 ALPHA-SUBSTITUTED ARYLMETHYL PIPERAZINE PYRAZOLO[1,5-α]PYRIMIDINE AMIDE DERIVATIVES PANACOS PHARMACEUTICALS, INC. (US) 2008-11-06 WO disclosed
WO-2008134035-A1 ALPHA-UNSUBSTITUTED ARYLMETHYL PIPERAZINE PYRAZOLO[1,5-A] PYRIMIDINE AMIDE DERIVATIVES PANACOS PHARMACEUTICALS, INC. (US) 2008-11-06 WO disclosed
WO-2007137874-A2 IMIDAZOLIDINE DERIVATIVES, USES THEREFOR, PREPARATION THEREOF AND COMPOSITIONS COMPRISING SUCH GALAPAGOS SAS (FR) 2007-12-06 WO disclosed