Flumethasone

Flumethasone

SCHEMBL4046

C[C@@H]1C[C@H]2[C@@H]3C[C@H](F)C4=CC(=O)C=C[C@]4(C)[C@@]3(F)[C@@H](O)C[C@]2(C)[C@@]1(O)C(=O)CO

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 7/20 1.00
PGR P06401 6/20 1.00
AR P10275 6/20 1.00
HIF1A Q16665 5/20 1.00
MAPT P10636 2/20 1.00
ABCB11 O95342 1/20 1.00
ALDH1A1 P00352 1/20 1.00
RAB9A P51151 1/20 1.00
SMN1; SMN2 Q16637 1/20 1.00
NR3C1 P04150 9/20 0.76
GAA P10253 1/20 0.75
CHRM1 P11229 1/20 0.75
TBXA2R P21731 1/20 0.75
ADRA1A P35348 1/20 0.75
HSD17B10 Q99714 3/20 0.71
TSHR P16473 2/20 0.71
NFKB1 P19838 2/20 0.71
MEN1 O00255 1/20 0.71
CYP2D6 P10635 1/20 0.71
KMT2A Q03164 1/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Flumethasone SCHEMBL4555 1.00 CYP3A4 (1.00) CYP3A4PGRARHIF1AMAPT
Flumethasone SCHEMBL3167856 1.00 CYP3A4 (1.00) CYP3A4PGRARHIF1AMAPT
Flumethasone SCHEMBL13046613 1.00 CYP3A4 (1.00) CYP3A4PGRARHIF1AMAPT
Flumethasone SCHEMBL11123357 1.00 CYP3A4 (1.00) CYP3A4PGRARHIF1AMAPT
Flumethasone SCHEMBL11844543 1.00 CYP3A4 (1.00) CYP3A4PGRARHIF1AMAPT
Flumethasone SCHEMBL10422222 1.00 CYP3A4 (1.00) CYP3A4PGRARHIF1AMAPT
Flumethasone SCHEMBL11911307 1.00 CYP3A4 (1.00) CYP3A4PGRARHIF1AMAPT
Flumethasone SCHEMBL3167846 1.00 CYP3A4 (1.00) CYP3A4PGRARHIF1AMAPT
Flumethasone SCHEMBL9910827 1.00 CYP3A4 (1.00) CYP3A4PGRARHIF1AMAPT
Flumethasone SCHEMBL20169795 1.00 CYP3A4 (1.00) CYP3A4PGRARHIF1AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 12369 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026100654-A1 NUCLEIC ACID INTRODUCTION AID, NUCLEIC ACID INTRODUCTION AGENT, AND NUCLEIC ACID INTRODUCTION METHOD 株式会社インファーマシア 2026-05-15 WO claimed
EP-4736841-A1 A MUCOADHESIVE LAYER FOR BUCCAL ADMINISTRATION OF AN ACTIVE PHARMACEUTICAL INGREDIENT IQ medical GmbH (DE) 2026-05-06 EP claimed
EP-4722714-A1 SIMULTANEOUS ANALYSIS OF FOOD-BORNE DOPING SUBSTANCES USING LIQUID CHROMATOGRAPHY-MASS SPECTROMETRY (VFD: VACCINE FOR FOODBORNE DOPING) Korea Institute of Science and Technology (KR) 2026-04-08 EP claimed
EP-4683679-A1 METHOD FOR DIAGNOSING AND TREATING NIS-EXPRESSING CARCINOMAS AND METASTASES NUSKE, Andreas (DE) 2026-01-28 EP claimed
EP-4301343-B1 PHARMACEUTICAL COMPOSITIONS WITH REDUCED SIDE EFFECT AND METHODS OF USING THE SAME TLC BIOPHARMACEUTICALS INC (US) 2025-11-19 EP claimed
US-20250255781-A1 PROCESSES FOR PREPARATION OF 3-D PRINTED PHARMACEUTICAL PRODUCTS BRISTOL-MYERS SQUIBB COMPANY (US) 2025-08-14 US claimed
US-12377144-B2 Methods of treating cancer using multi-specific binding proteins that bind NKG2D, CD16 and a tumor-associated antigen DRAGONFLY THERAPEUTICS, INC. (US) 2025-08-05 US claimed
US-20250205227-A1 METHODS FOR ADMINISTERING CORTICOSTEROIDS SPARROW PHARMACEUTICALS, INC. 2025-06-26 US claimed
WO-2025123147-A1 TOLERIZING IMMUNOMODULATORY COMBINATION INTEGRATED NANOTHERAPEUTICS INC. (CA) 2025-06-19 WO claimed
US-20250186365-A1 COMBINATION OF ANTISPASMODIC AND OSMOTIC AGENTS FOR TOPICAL PRODUCTS AND METHOD OF USE THEREOF PRIMA INNOVATIONS, LLC 2025-06-12 US claimed
EP-0055870-A1 Pyridylmethyl esters of selected bio-affecting carboxylic acids, process for preparing and pharmaceutical composition comprising the same MERCK & CO. INC. (US) 1982-07-14 EP claimed
US-4333927-A CORTICOSTEROID, PHOSPHATIDE, BUTYLHYDROXYANISOLE AND/OR BUTYLHYDROXYTOLUENE MITSUBISHI CHEMICAL INDUSTRIES, LTD. (JP) 1982-06-08 US claimed
EP-0051278-A1 Soft tertiary amine esters of bio-affecting carboxylic acids, processes for preparing and a pharmaceutical composition containing the same MERCK & CO. INC. (US) 1982-05-12 EP claimed
US-4279900-A ANTIINFLAMMATORY INTREX RESEARCH CORPORATION (US) 1981-07-21 US claimed
EP-0028110-A2 Autoclavable emulsions Smith and Nephew Associated Companies p.l.c. (GB) 1981-05-06 EP claimed
US-4244942-A Creamy preparation containing steroid and process for the preparation thereof TOKO YAKUHIN KOGYO KABUSHIKI KAISHA (JP) 1981-01-13 US claimed
US-4221787-A Esteramide prodrugs of anti-inflammatory corticosteroids INTERX RESEARCH CORPORATION (US) 1980-09-09 US claimed
US-4112073-A Medicinal composition comprising adrenal cortical hormone and thyroid stimulating hormone releasing hormone TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1978-09-05 US claimed
US-4083974-A Topical steroidal anti-inflammatory preparations containing polyoxypropylene 15 stearyl ether THE UPJOHN COMPANY (US) 1978-04-11 US claimed
US-4041055-A SULFENYLATION, MICHAEL ADDITION, REACTION WITH THIOPHILE, HYDROLYSIS THE UPJOHN COMPANY (US) 1977-08-09 US claimed