Flumethasone

Flumethasone

SCHEMBL4555

C[C@H]1C[C@H]2[C@@H]3C[C@H](F)C4=CC(=O)C=C[C@]4(C)[C@@]3(F)[C@@H](O)C[C@]2(C)[C@@]1(O)C(=O)CO

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 7/20 1.00
PGR P06401 6/20 1.00
AR P10275 6/20 1.00
HIF1A Q16665 5/20 1.00
MAPT P10636 2/20 1.00
ABCB11 O95342 1/20 1.00
ALDH1A1 P00352 1/20 1.00
RAB9A P51151 1/20 1.00
SMN1; SMN2 Q16637 1/20 1.00
NR3C1 P04150 9/20 0.76
GAA P10253 1/20 0.75
CHRM1 P11229 1/20 0.75
TBXA2R P21731 1/20 0.75
ADRA1A P35348 1/20 0.75
HSD17B10 Q99714 3/20 0.71
TSHR P16473 2/20 0.71
NFKB1 P19838 2/20 0.71
MEN1 O00255 1/20 0.71
CYP2D6 P10635 1/20 0.71
KMT2A Q03164 1/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Flumethasone SCHEMBL3167856 1.00 CYP3A4 (1.00) CYP3A4PGRARHIF1AMAPT
Flumethasone SCHEMBL13046613 1.00 CYP3A4 (1.00) CYP3A4PGRARHIF1AMAPT
Flumethasone SCHEMBL11123357 1.00 CYP3A4 (1.00) CYP3A4PGRARHIF1AMAPT
Flumethasone SCHEMBL11844543 1.00 CYP3A4 (1.00) CYP3A4PGRARHIF1AMAPT
Flumethasone SCHEMBL10422222 1.00 CYP3A4 (1.00) CYP3A4PGRARHIF1AMAPT
Flumethasone SCHEMBL11911307 1.00 CYP3A4 (1.00) CYP3A4PGRARHIF1AMAPT
Flumethasone SCHEMBL4046 1.00 CYP3A4 (1.00) CYP3A4PGRARHIF1AMAPT
Flumethasone SCHEMBL3167846 1.00 CYP3A4 (1.00) CYP3A4PGRARHIF1AMAPT
Flumethasone SCHEMBL9910827 1.00 CYP3A4 (1.00) CYP3A4PGRARHIF1AMAPT
Flumethasone SCHEMBL20169795 1.00 CYP3A4 (1.00) CYP3A4PGRARHIF1AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 10461 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260137656-A1 METHODS AND COMPOSITIONS FOR TREATING GLUCOCORTICOID EXCESS SPARROW PHARMACEUTICALS INC (US) 2026-05-21 US claimed
US-20260137657-A1 METHODS AND COMPOSITIONS FOR TREATING GLUCOCORTICOID EXCESS SPARROW PHARMACEUTICALS INC (US) 2026-05-21 US claimed
EP-4744657-A1 THERAPEUTIC AGENT FOR HUMAN GRAFT VERSUS HOST DISEASE AND COMBINATION THEREOF National University Corporation Okayama University (JP) 2026-05-20 EP claimed
WO-2026100654-A1 NUCLEIC ACID INTRODUCTION AID, NUCLEIC ACID INTRODUCTION AGENT, AND NUCLEIC ACID INTRODUCTION METHOD 株式会社インファーマシア 2026-05-15 WO claimed
US-20260027255-A1 Cross-Linked Telechelic Polymer Compositions, Methods of Preparation Thereof, and Methods of Using Same BETTY YU SKIN TECH ADVISORS LLC (US) 2026-01-29 US claimed
US-20250319104-A1 MOISTURIZING CREAM FOR RADIATION DERMATITIS PERRY ARTHUR W (US) 2025-10-16 US claimed
US-20250302917-A1 METHODS OF REDUCING THE SIGNS OR SYMPTOMS OF DERMAL DISORDERS WITH TOPICALLY APPLIED SILK FIBROIN COCOON BIOTECH INC (US) 2025-10-02 US claimed
US-20250288585-A1 SYNERGISTIC COMPOSITIONS FOR ENHANCED HAIR GROWTH AND METHODS FOR TREATING HAIR LOSS THE JOHNS HOPKINS UNIVERSITY 2025-09-18 US claimed
EP-4615506-A1 USE OF GSK-3 ACTIVATIOR TO MODULATE PROTEASOME ACTIVITY TO PREVENT AGEING ASSOCIATED CONDITIONS AND DISEASES Sahin, Fikret (TR) 2025-09-17 EP claimed
US-20250255781-A1 PROCESSES FOR PREPARATION OF 3-D PRINTED PHARMACEUTICAL PRODUCTS BRISTOL-MYERS SQUIBB COMPANY (US) 2025-08-14 US claimed
US-5049387-A Inducing skin tolerance to a sensitizing drug ALZA CORPORATION (US) 1991-09-17 US claimed
US-5036048-A Angiotensin II receptor blockers as antiglaucoma agents SCHERING CORPORATION (US) 1991-07-30 US claimed
US-5017567-A Steroid antiinflammatory SCHERING CORPORATION (US) 1991-05-21 US claimed
US-4885293-A CARBOXYALKYL DIPEPTIDES SCHERING CORPORATION (US) 1989-12-05 US claimed
US-4840772-A KIT WITH CONTAINERS OF AGENT TO REDUCE INTRAOCULAR PRESSURE AND ANTIINFLAMMATORY STEROID OR BETA-BLOCKER SCHERING CORPORATION (US) 1989-06-20 US claimed
EP-0186948-B1 PROCESS AND INTERMEDIATES FOR THE PREPARATION OF 17ALPHA-HYDROXYPROGESTERONES AND CORTICOIDS FROM AN ENOL STEROID THE UPJOHN COMPANY (US) 1989-01-25 EP claimed
US-4783444-A SUBSTITUTED DIPEPTIDES SCHERING CORPORATION (US) 1988-11-08 US claimed
EP-0186948-A1 Process and intermediates for the preparation of 17alpha-hydroxyprogesterones and corticoids from an enol steroid THE UPJOHN COMPANY (US) 1986-07-09 EP claimed
EP-0068553-B1 TOPICAL ANTIMICROBIAL ANTI-INFLAMMATORY COMPOSITIONS THE PROCTER & GAMBLE COMPANY (US) 1985-11-21 EP claimed
US-3980778-A Anti-inflammatory steroid THE UPJOHN COMPANY (US) 1976-09-14 US claimed